SCHEMBL425964

SCHEMBL425964

[CH2]C(=O)N1CCC(N(C)C)CC1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL3 Q96JM7 2/20 0.56
L3MBTL1 Q9Y468 1/20 0.45
CDYL Q9Y232 1/20 0.38
CDY1; CDY1B Q9Y6F8 1/20 0.38
HDAC4 P56524 1/20 0.36
KDM1A O60341 3/20 0.34
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
PARP1 P09874 2/20 0.34
MCHR1 Q99705 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.33
USP5 P45974 1/20 0.32
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
MALT1 Q9UDY8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1196738 0.88 L3MBTL3 (0.49) L3MBTL3L3MBTL1KDM1AMAOAMAOB
SCHEMBL27781047 0.82 L3MBTL3 (0.60) L3MBTL3L3MBTL1CDYLCDY1; CDY1BHDAC4
SCHEMBL4550247 0.80 L3MBTL3 (0.58) L3MBTL3L3MBTL1SMN1; SMN2
SCHEMBL3104303 0.80 L3MBTL3 (0.58) L3MBTL3L3MBTL1CDYLCDY1; CDY1BHDAC4
SCHEMBL8362221 0.78 L3MBTL3 (0.56) L3MBTL3L3MBTL1CDYLCDY1; CDY1BHDAC4
SCHEMBL20842232 0.78 L3MBTL3 (0.56) L3MBTL3L3MBTL1CDYLCDY1; CDY1BHDAC4
SCHEMBL3068209 0.78 L3MBTL3 (0.56) L3MBTL3L3MBTL1CDYLCDY1; CDY1BHDAC4
SCHEMBL22878132 0.78 L3MBTL3 (0.56) L3MBTL3L3MBTL1CDYLCDY1; CDY1BHDAC4
SCHEMBL3940873 0.78 ACKR3 (0.43) L3MBTL3L3MBTL1CDYLCDY1; CDY1BMEN1
SCHEMBL31387583 0.78 L3MBTL3 (0.51) L3MBTL3L3MBTL1CDYLCDY1; CDY1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2011524411-A 2011-09-01 JP claimed
CN-102124000-A Pyridine compounds ASTRAZENECA AB 2011-07-13 CN claimed
US-20110166139-A1 PYRIDINE COMPOUNDS ASTRAZENECA AB (SE) 2011-07-07 US claimed
EP-2303861-A1 PYRIDINE COMPOUNDS AstraZeneca AB (SE) 2011-04-06 EP claimed
WO-2009153589-A1 PYRIDINE COMPOUNDS ASTRAZENECA AB (SE) 2009-12-23 WO claimed
EP-2044083-A1 ANTIVIRAL AGENTS GENELABS TECHNOLOGIES, INC. (US) 2009-04-08 EP claimed
US-20080051384-A1 ANTIVIRAL AGENTS GENELABS TECHNOLOGIES, INC. 2008-02-28 US claimed
WO-2008008912-A1 ANTIVIRAL AGENTS GENELABS TECHNOLOGIES, INC. (US) 2008-01-17 WO claimed
WO-2008008907-A2 ANTIVIRAL AGENTS GENELABS TECHNOLOGIES, INC. (US) 2008-01-17 WO claimed
EP-1844042-A1 INDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2007-10-17 EP claimed
US-20060211698-A1 Bicyclic heteroaryl derivatives for treating viruses GENELABS, INC. 2006-09-21 US claimed
WO-2006076529-A1 INDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2006-07-20 WO claimed
CN-1077891-C 5-phenyl-3- (piperidin-4-yl) -1,3, 4-oxadiazol-2 (3H) -one derivatives useful as 5-HT4 or H3 receptor ligands SYNTHELABO (FR) 2002-01-16 CN claimed
US-5929089-A ANTISEROTONINE AGENT SYNTHELABO (FR) 1999-07-27 US claimed
EP-0863897-B1 5-PHENYL-3-(PIPERIDIN-4-YL)-1,3,4-OXADIAZOL-2(3H)-ONE DERIVATIVES FOR USE AS 5-HT4- OR H3-RECEPTOR LIGANDS SYNTHELABO (FR) 1999-06-16 EP claimed
CN-1202169-A 5-phenyl-3- (piperidin-4-yl) -1, 3, 4-oxadiazol-2 (3H) -one derivatives useful as 5-HT 4 or H3 receptor ligands SYNTHELABO (FR) 1998-12-16 CN claimed
CN-102124000-B Pyridine compounds ASTRAZENECA AB 2014-09-17 CN disclosed
EP-2303861-B1 PYRIDINE COMPOUNDS ASTRAZENECA AB (SE) 2014-04-23 EP disclosed
WO-2006076529-A1 INDOLE DERIVATIVES FOR TREATING VIRAL INFECTIONS GENELABS TECHNOLOGIES, INC. (US) 2006-07-20 WO disclosed
US-5929089-A ANTISEROTONINE AGENT SYNTHELABO (FR) 1999-07-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060211698-A1 Bicyclic heteroaryl derivatives for treating viruses HAVCR2, ZC3HAV1, SARS1 L3MBTL3 1385/4885L3MBTL1 1887/4885CDYL 1986/4885
US-20110166139-A1 PYRIDINE COMPOUNDS PTK2, PTK2B, PFKP L3MBTL3 4396/4885L3MBTL1 4279/4885CDYL 1611/4885
US-20080051384-A1 ANTIVIRAL AGENTS EIF2AK2, MAVS, ZC3HAV1 L3MBTL3 2698/4885L3MBTL1 3239/4885CDYL 4218/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.