SCHEMBL4263897

SCHEMBL4263897

O=S(=O)(c1ccccc1)c1cc2cc(O)c(F)cc2[nH]1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.40
HTR6 P50406 2/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
GFER P55789 1/20 0.39
DAO P14920 3/20 0.37
DDO Q99489 2/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA7 P43166 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
AKR1B1 P15121 2/20 0.35
CNR1 P21554 1/20 0.35
FEN1 P39748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27867018 0.78 KDM4E (0.47) CA2HTR6DAOKDM4EALDH1A1
SCHEMBL31561597 0.75 CA2 (0.62) CA2HTR6DAOCA12CA1
SCHEMBL3237494 0.75 CA2 (0.62) CA2HTR6DAOCA12CA1
SCHEMBL27462488 0.72 HRH3 (0.44) CA2HTR6DAOKDM4EAKR1B1
SCHEMBL17803693 0.72 CA2 (0.42) CA2HTR6CA1AKR1B1CNR1
SCHEMBL7407839 0.72 CNR1 (0.54) CA2HTR6AKR1B1CNR1
SCHEMBL6618503 0.72 CA2 (0.46) CA2HTR6KDM4EALDH1A1AKR1B1
SCHEMBL5190594 0.72 AKR1B1 (0.56) CA2HTR6DAOKDM4EALDH1A1
SCHEMBL8960443 0.72 HTR6 (0.56) CA2HTR6POLBGAAGFER
SCHEMBL8120975 0.72 KDM4E (0.49) CA2HTR6POLBDAOCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091953-A1 8-SULFONYL-L, 3, 4, 8-TETRAHYDR0-2H- [1, 4]OXAZEPINO [6, 7-E]INDOLE DERIVATIVES AND THEIR USE AS 5-HT6 RECEPTOR LIGANDS BIOVITRUM AB (publ) (SE) 2009-08-26 EP disclosed
WO-2008054288-A1 8-SULFONYL-L, 3, 4, 8-TETRAHYDR0-2H- [1, 4] OXAZEPINO [6, 7-E] INDOLE DERIVATIVES AND THEIR USE AS 5-HT6 RECEPTOR LIGANDS BIOVITRUM AB (PUBL) (SE) 2008-05-08 WO disclosed