SCHEMBL4264289

SCHEMBL4264289

Cn1c(NCCO)nc(=O)c2c1ncn2Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.54
ADORA2B P29275 1/20 0.54
RXFP1 Q9HBX9 1/20 0.54
ALDH1A1 P00352 2/20 0.53
PCSK9 Q8NBP7 1/20 0.53
POLB P06746 2/20 0.49
HIF1A Q16665 1/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 2/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 3/20 0.47
TP53 P04637 2/20 0.45
PDE1A P54750 1/20 0.45
PDE1B Q01064 1/20 0.45
PDE1C Q14123 1/20 0.45
P2RX7 Q99572 3/20 0.44
THRB P10828 1/20 0.43
GLA P06280 1/20 0.43
UBE2N P61088 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7445594 0.82 SMN1; SMN2 (0.62) SMN1; SMN2ADORA2BRXFP1ALDH1A1PCSK9
SCHEMBL4263443 0.78 SMN1; SMN2 (0.64) SMN1; SMN2ADORA2BRXFP1ALDH1A1POLB
SCHEMBL7443156 0.76 SMN1; SMN2 (0.54) SMN1; SMN2ADORA2BRXFP1ALDH1A1PCSK9
SCHEMBL7110383 0.71 SMN1; SMN2 (0.54) SMN1; SMN2ADORA2BRXFP1ALDH1A1POLB
SCHEMBL1944405 0.71 ADORA2B (1.00) SMN1; SMN2ADORA2BRXFP1ALDH1A1POLB
SCHEMBL555404 0.70 PDE1A (0.73) SMN1; SMN2ADORA2BRXFP1ALDH1A1POLB
SCHEMBL8179399 0.70 SMN1; SMN2 (0.49) SMN1; SMN2ADORA2BRXFP1ALDH1A1POLB
SCHEMBL12604460 0.70 PCSK9 (1.00) SMN1; SMN2ALDH1A1PCSK9MEN1KMT2A
SCHEMBL20011033 0.69 SMN1; SMN2 (0.76) SMN1; SMN2ADORA2BRXFP1ALDH1A1POLB
SCHEMBL9586511 0.69 PCSK9 (0.51) SMN1; SMN2ALDH1A1PCSK9POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009144548-A1 IMIDAZO [2,1-B] PURINE DERIVATIVES AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2009-12-03 WO disclosed