SCHEMBL4270776

SCHEMBL4270776

O=C(O)/C=C/C1=Cc2ccccc2CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.44
HDAC3 O15379 1/20 0.44
TNKS O95271 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
MITF O75030 1/20 0.40
HSP90AA1 P07900 1/20 0.40
RAB9A P51151 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4264349 1.00 HCAR2 (0.44) HCAR2HDAC3TNKSHDAC4HDAC1
Pyrrole SCHEMBL4268503 0.91 HDAC3 (0.38) HCAR2HDAC3TNKSHDAC4HDAC1
SCHEMBL4264341 0.85 MEN1 (0.47) RAB9AKDM4EALDH1A1HPGDGPR183
SCHEMBL4268501 0.79 GPR183 (0.49) RAB9AKDM4EALDH1A1HPGDGPR183
SCHEMBL2531349 0.79 GPR84 (0.41) MAOAMAOBPTGS2CYP19A1CYP11B1
SCHEMBL2531348 0.79 GPR84 (0.41) MAOAMAOBPTGS2CYP19A1CYP11B1
SCHEMBL4266852 0.78 TRPM8 (0.36) PTGS1PTGS2GPR183KDM1ALMNA
SCHEMBL4276499 0.78 NPC1 (0.52) RAB9AALDH1A1MAOAMAOBPTGS1
SCHEMBL4266849 0.78 TRPM8 (0.36) PTGS1PTGS2GPR183KDM1ALMNA
SCHEMBL4276500 0.78 NPC1 (0.52) RAB9AALDH1A1MAOAMAOBPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110002-A1 NOVEL EFFLUX PUMP INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-11 WO claimed
WO-2009110002-A1 NOVEL EFFLUX PUMP INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-11 WO disclosed