Pyrrole

Pyrrole

SCHEMBL4268503

O=C(O)C=CC1=Cc2ccccc2CC1.c1cc[nH]c1

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.38
TNKS O95271 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
CYP3A4 P08684 1/20 0.36
RECQL P46063 1/20 0.36
PMP22 Q01453 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4270776 0.91 HCAR2 (0.44) HDAC3TNKSHDAC4HDAC1HCAR2
SCHEMBL4264349 0.91 HCAR2 (0.44) HDAC3TNKSHDAC4HDAC1HCAR2
SCHEMBL4264341 0.78 MEN1 (0.47) MEN1KMT2ARAB9AKDM4EALDH1A1
Pyrrole SCHEMBL4270409 0.77 ALDH1A1 (0.40) MEN1LMNAKMT2AKDM4EALDH1A1
SCHEMBL4276499 0.74 NPC1 (0.52) RAB9AALDH1A1PTGS1PTGS2MAOA
SCHEMBL4276500 0.74 NPC1 (0.52) RAB9AALDH1A1PTGS1PTGS2MAOA
SCHEMBL4266849 0.74 TRPM8 (0.36) MEN1LMNACYP3A4RECQLPMP22
SCHEMBL4266852 0.74 TRPM8 (0.36) MEN1LMNACYP3A4RECQLPMP22
SCHEMBL4268501 0.72 GPR183 (0.49) MEN1LMNAKMT2ARAB9AKDM4E
SCHEMBL2531349 0.72 GPR84 (0.41) PTGS2MAOAMAOBGPR183

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110002-A1 NOVEL EFFLUX PUMP INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-11 WO claimed
WO-2009110002-A1 NOVEL EFFLUX PUMP INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-11 WO disclosed