SCHEMBL42757

SCHEMBL42757

O=Cc1ccc(F)c(Cl)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.64
HSD17B10 Q99714 1/20 0.52
ALDH1A3 P47895 3/20 0.48
VCAM1 P19320 1/20 0.46
ALDH3A1 P30838 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
TRPA1 O75762 1/20 0.42
TTR P02766 1/20 0.42
KDM4E B2RXH2 1/20 0.41
PTGS2 P35354 1/20 0.41
RAB9A P51151 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
KIF11 P52732 1/20 0.39
SLC2A1 P11166 1/20 0.39
PTGER4 P35408 1/20 0.39
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29472390 1.00 ALDH1A1 (0.64) ALDH1A1HSD17B10ALDH1A3VCAM1ALDH3A1
Hydrochloric Acid SCHEMBL30783012 0.98 ALDH1A1 (0.61) ALDH1A1HSD17B10ALDH1A3VCAM1ALDH3A1
SCHEMBL2009103 0.84 KIF11 (0.54) ALDH1A1HSD17B10PTGS2KIF11
SCHEMBL18002915 0.83 AHR (0.46) ALDH1A1HSD17B10ALDH1A3TRPA1KMT2A
SCHEMBL4847293 0.83 ALDH1A1 (0.46) ALDH1A1HSD17B10ALDH1A3VCAM1ALDH3A1
SCHEMBL190947 0.82 ALDH1A1 (0.64) ALDH1A1HSD17B10ALDH1A3VCAM1ALDH3A1
SCHEMBL8698264 0.80 ALDH1A1 (0.43) ALDH1A1TTRKDM4EPTGS2RAB9A
SCHEMBL18345531 0.79 XDH (0.48) ALDH1A1HSD17B10TRPA1KDM4ESLC2A1
SCHEMBL14989926 0.79 XDH (0.48) ALDH1A1HSD17B10TRPA1KDM4ESLC2A1
SCHEMBL3926234 0.79 HSD17B10 (0.45) ALDH1A1HSD17B10ALDH1A3VCAM1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1160 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118598815-A 2-Urea (thiourea) base-4-phenyl substituted quinazoline compound and preparation method and application thereof 西华大学 2024-09-06 CN claimed
CN-118496215-A Polyhydroxylated onium derivative with disubstituted benzene ring, preparation method and medical application thereof 中国药科大学 2024-08-16 CN claimed
CN-117624148-A Polyhydroxy sulfonium salt derivative with disubstituted benzene ring, preparation method and medical application thereof 中国药科大学 2024-03-01 CN claimed
CN-112266352-B Piperlongumine derivative and preparation method and application thereof 绍兴文理学院 2022-02-08 CN claimed
CN-112266352-A Piperlongumine derivative and preparation method and application thereof 绍兴文理学院 2021-01-26 CN claimed
US-RE48335-E1 Polymyxin derivatives as antimicrobial compounds MONASH UNIVERSITY (AU) 2020-12-01 US claimed
CN-106414480-B Polymyxin derivatives as antimicrobial compounds 莫纳什大学 2020-08-04 CN claimed
CN-107188851-B Method for synthesizing astemizole key intermediate and derivative thereof 湖南大学 2020-04-07 CN claimed
US-20180273906-A1 MICROVESICLE AND STEM CELL COMPOSITIONS FOR THERAPEUTIC APPLICATIONS IPS HEART 2018-09-27 US claimed
US-10017684-B2 Method and compositions for hydraulic fracturing and for tracing formation water SPECTRUM TRACER SERVICES, LLC (US) 2018-07-10 US claimed
EP-1773843-A4 SMALL MOLECULE THIENOPYRIMIDINE-BASED PROTEIN TYROSINE KINASE INHIBITORS UNIV TEXAS (US) 2009-06-03 EP claimed
EP-1773843-A1 SMALL MOLECULE THIENOPYRIMIDINE-BASED PROTEIN TYROSINE KINASE INHIBITORS The Board of Regents of The University of Texas System (US) 2007-04-18 EP claimed
US-20060084176-A1 Detection of uronium salts YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2006-04-20 US claimed
WO-2006014404-A1 SMALL MOLECULE THIENOPYRIMIDINE-BASED PROTEIN TYROSINE KINASE INHIBITORS BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2006-02-09 WO claimed
US-20060004002-A1 Small molecule thienopyrimidine-based protein tyrosine kinase inhibitors BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2006-01-05 US claimed
EP-0979812-B1 Process for the preparation of fluorinated benzyl alcools and benzyl aldehydes BAYER AG (DE) 2003-10-29 EP claimed
EP-0903334-B1 Halogenated aromatic derivatives and process for the preparation thereof MITENI SPA (IT) 2003-06-11 EP claimed
EP-0922693-B1 Process for the preparation of 3-chloro-4-fluorobenzoyl chloride CLARIANT GMBH (DE) 2001-10-24 EP claimed
US-6127581-A Process for preparing fluorinated benzyl alcohols and fluorinated benzaldehydes BAYER AKTIENGESELLSCHAFT (DE) 2000-10-03 US claimed
EP-0979812-A1 Process for the preparation of fluorinated benzyl alcools and benzyl aldehydes Bayer Aktiengesellschaft (DE) 2000-02-16 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004002-A1 Small molecule thienopyrimidine-based protein tyrosine kinase inhibitors SRC, LCK, FYN ALDH1A1 4583/4885HSD17B10 4240/4885ALDH1A3 4871/4885
US-20180273906-A1 MICROVESICLE AND STEM CELL COMPOSITIONS FOR THERAPEUTIC APPLICATIONS EXOSC9, EXOSC5, EXOSC4 ALDH1A1 493/4885HSD17B10 3195/4885ALDH1A3 872/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.