SCHEMBL4282256

SCHEMBL4282256

COC(=O)N1CCCC(c2ccc(F)cc2C)C1N

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 7/20 0.43
TACR1 P25103 3/20 0.41
NPSR1 Q6W5P4 1/20 0.40
GRM5 P41594 2/20 0.38
OPRL1 P41146 2/20 0.38
RIPK1 Q13546 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
CHRM3 P20309 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4285494 0.83 SLC6A3 (0.43)
SCHEMBL4291883 0.80 SLC6A3 (0.46) NPSR1RIPK1KDM4ELMNACHRM3
SCHEMBL4280120 0.80 LMNA (0.40) HCRTR2NPSR1LMNA
SCHEMBL4282253 0.79 TACR1 (0.41) HCRTR2TACR1NPSR1GRM5OPRL1
SCHEMBL4291624 0.77 HCRTR2 (0.42) HCRTR2NPSR1
SCHEMBL4288939 0.76 TSHR (0.44) NPSR1LMNA
SCHEMBL4285849 0.75 SLC6A4 (0.47) HCRTR2
SCHEMBL4281409 0.74 ALDH1A1 (0.38) NPSR1KDM4ELMNA
SCHEMBL4294072 0.73 CHRNB4 (0.41) HCRTR2
SCHEMBL4282512 0.73 HCRTR2 (0.47) HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009072643-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-11 WO disclosed