SCHEMBL4287682

SCHEMBL4287682

Nc1c[nH]nc1C(=O)NCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
GAA P10253 1/20 0.52
ADORA2A P29274 3/20 0.52
NSD2 O96028 2/20 0.50
KMT2A Q03164 2/20 0.49
ADORA1 P30542 2/20 0.48
PIN1 Q13526 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
HPGD P15428 1/20 0.47
MMP13 P45452 1/20 0.47
PKM P14618 2/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4279819 0.86 RAB9A (0.56) ALDH1A1ADORA2AKMT2AADORA1TSHR
SCHEMBL6500669 0.83 L3MBTL1 (0.57) ALDH1A1KMT2ACYP1A2CYP2C9TSHR
SCHEMBL13816854 0.83 ALDH1A1 (0.50) ALDH1A1GAAKMT2APIN1HPGD
SCHEMBL4289254 0.79 GAA (0.54) ALDH1A1GAAKMT2APIN1CYP1A2
SCHEMBL5274230 0.78 HPGD (0.49) ALDH1A1GAAKMT2AHPGD
SCHEMBL4284499 0.78 TDP1 (0.53) ALDH1A1ADORA2AKMT2AADORA1TSHR
SCHEMBL12245094 0.76 CCNE2 (0.40) ALDH1A1PIN1TSHRHPGD
SCHEMBL5274493 0.76 ALDH1A1 (0.46) ALDH1A1GAAADORA2AKMT2APIN1
SCHEMBL5268993 0.76 ALDH1A1 (0.54) ALDH1A1GAAKMT2ATSHRHPGD
SCHEMBL5268485 0.75 KCNA5 (0.51) ALDH1A1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090156582-A1 Pyrazole Compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-18 US disclosed
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156582-A1 Pyrazole Compound GSK3B, GSK3A, GSKIP ALDH1A1 694/4885GAA 2871/4885ADORA2A 1801/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.