SCHEMBL4289696

SCHEMBL4289696

Cc1ncccc1C(=O)Nc1c[nH]nc1C(=O)NC1CCCC1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 1/20 0.49
GAA P10253 1/20 0.49
RAB9A P51151 3/20 0.47
ACKR3 P25106 1/20 0.46
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
PKM P14618 1/20 0.44
CNR2 P34972 4/20 0.43
CNR1 P21554 3/20 0.43
HSD11B1 P28845 1/20 0.43
HTT P42858 1/20 0.43
NPC1 O15118 2/20 0.43
P2RX7 Q99572 1/20 0.42
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4292724 0.88 CNR2 (0.49) ALDH1A1KDM4EGAARAB9AACKR3
SCHEMBL4282985 0.82 GRM5 (0.56) ALDH1A1KDM4EGAARAB9APKM
SCHEMBL4292371 0.81 GRM5 (0.55) ALDH1A1KDM4EGAARAB9AACKR3
SCHEMBL4285069 0.80 ACKR3 (0.45) ALDH1A1RAB9AACKR3CYP1A2CYP2C19
SCHEMBL5269272 0.78 KDM4E (0.55) ALDH1A1KDM4ERAB9AMEN1KMT2A
SCHEMBL5268963 0.78 LMNA (0.46) ALDH1A1RAB9AMEN1CYP1A2CYP3A4
SCHEMBL5265256 0.77 RAB9A (0.57) ALDH1A1RAB9AACKR3MEN1KMT2A
SCHEMBL12709415 0.76 P2RX7 (0.61) ALDH1A1KDM4EGAARAB9AMEN1
SCHEMBL4288778 0.76 CDK2 (0.61) RAB9AACKR3MEN1KMT2APKM
SCHEMBL4281636 0.76 PTGES (0.47) ALDH1A1KDM4EGAARAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090156582-A1 Pyrazole Compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-18 US disclosed
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156582-A1 Pyrazole Compound GSK3B, GSK3A, GSKIP ALDH1A1 694/4885KDM4E 810/4885GAA 2871/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.