SCHEMBL4292183

SCHEMBL4292183

O=c1ccc2ccncc2n1F

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPT P10636 14/20 0.38
CYP19A1 P11511 2/20 0.38
DAO P14920 1/20 0.36
CDC7 O00311 1/20 0.36
CDK2 P24941 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
RAPGEF4 Q8WZA2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8268970 0.77 BRPF1 (0.55) MAPTCYP19A1CDC7CDK2
SCHEMBL30833284 0.77 BRPF1 (0.55) MAPTCYP19A1CDC7CDK2
SCHEMBL28855321 0.72 HDAC1 (0.38) MAPTCYP19A1
SCHEMBL1054493 0.71 CA12 (0.57) MAPTDAO
SCHEMBL4133896 0.70 CDK4 (0.37) MAPTCYP19A1DAOCDC7CDK2
SCHEMBL12065990 0.69 KDM4E (0.47)
SCHEMBL4128204 0.66 CDK4 (0.34) MAPTCYP19A1DAORAPGEF4
SCHEMBL4755903 0.65 DAO (0.43) DAOCDC7CDK2PDE3BPDE3A
SCHEMBL2614351 0.65 BRPF1 (0.55) MAPTCDC7CDK2PDE3BPDE3A
SCHEMBL30066887 0.65 BRPF1 (0.55) MAPTCDC7CDK2PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090281100-A1 Benzimidazole quinolinones and uses thereof BARSANTI PAUL A 2009-11-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090281100-A1 Benzimidazole quinolinones and uses thereof GAA, ALPI, IL4I1 MAPT 575/4885CYP19A1 868/4885DAO 371/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.