SCHEMBL4301494

SCHEMBL4301494

COC(=O)c1cc(O)cn1CC(=O)c1cccc(F)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.44
LMNA P02545 4/20 0.44
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
NPC1 O15118 5/20 0.43
KDM4E B2RXH2 4/20 0.43
MAPT P10636 4/20 0.43
RAB9A P51151 4/20 0.43
HPGD P15428 3/20 0.43
HTT P42858 3/20 0.43
TSHR P16473 2/20 0.43
ALOX12 P18054 1/20 0.43
SMN1; SMN2 Q16637 5/20 0.43
NPSR1 Q6W5P4 2/20 0.43
KCNH2 Q12809 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 2/20 0.42
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
GRIN2B Q13224 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313102 0.85 CDYL2 (0.52) LMNAKMT2AMEN1NPC1KDM4E
SCHEMBL4306365 0.85 LMNA (0.45) LMNAKMT2AMEN1KDM4EHPGD
SCHEMBL4306412 0.85 KMT2A (0.42) MRGPRX4LMNAKMT2AMEN1NPC1
SCHEMBL4305020 0.81 LMNA (0.46) LMNAKMT2AMEN1KDM4EMAPT
SCHEMBL4305068 0.81 LMNA (0.47) LMNAKMT2AMEN1NPC1KDM4E
SCHEMBL4311072 0.76 MRGPRX4 (0.37) MRGPRX4LMNAKMT2AMEN1NPC1
SCHEMBL4304270 0.75 CYP1A2 (0.43) LMNAKDM4EMAPTALDH1A1
SCHEMBL8015699 0.74 PKM (0.44) LMNAKMT2AMEN1NPC1KDM4E
SCHEMBL8022961 0.72 NPC1 (0.45) LMNAKMT2AMEN1NPC1KDM4E
SCHEMBL17070601 0.72 KMT2A (0.69) MRGPRX4LMNAKMT2AMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009130231-A1 PYRROLO [1, 2-A] PYRAZINE DERIVATIVES AS VASOPRESSIN VIB RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-10-29 WO disclosed
WO-2009130231-A1 PYRROLO [1, 2-A] PYRAZINE DERIVATIVES AS VASOPRESSIN VIB RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-10-29 WO disclosed