SCHEMBL4313102

SCHEMBL4313102

COC(=O)c1cc(O)cn1CC(=O)c1cccc(OC)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDYL2 Q8N8U2 4/20 0.52
CDYL Q9Y232 4/20 0.52
CDY1; CDY1B Q9Y6F8 4/20 0.52
NPC1 O15118 6/20 0.51
RAB9A P51151 6/20 0.51
SMN1; SMN2 Q16637 5/20 0.51
POLB P06746 2/20 0.51
BLM P54132 1/20 0.51
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
MAPT P10636 3/20 0.46
HPGD P15428 2/20 0.46
KDM4E B2RXH2 1/20 0.46
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
TP53 P04637 3/20 0.46
CBX7 O95931 2/20 0.46
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4306365 0.85 LMNA (0.45) POLBHPGDKDM4EMEN1KMT2A
SCHEMBL4301494 0.85 MRGPRX4 (0.44) NPC1RAB9ASMN1; SMN2POLBESR1
SCHEMBL4302800 0.85 CDYL2 (0.49) CDYL2CDYLCDY1; CDY1BNPC1RAB9A
SCHEMBL4307512 0.84 CDYL2 (0.48) CDYL2CDYLCDY1; CDY1BNPC1RAB9A
SCHEMBL8022961 0.80 NPC1 (0.45) CDYL2CDYLCDY1; CDY1BNPC1RAB9A
SCHEMBL4306740 0.77 KMT2A (0.59) POLBESR1MAPTKDM4EMEN1
SCHEMBL4305020 0.76 LMNA (0.46) MAPTHPGDKDM4EMEN1KMT2A
SCHEMBL8015699 0.74 PKM (0.44) NPC1RAB9ASMN1; SMN2POLBESR1
SCHEMBL11248287 0.73 CES2 (0.69) NPC1RAB9ASMN1; SMN2POLBBLM
SCHEMBL30758862 0.73 CES2 (0.69) NPC1RAB9ASMN1; SMN2POLBBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009130231-A1 PYRROLO [1, 2-A] PYRAZINE DERIVATIVES AS VASOPRESSIN VIB RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-10-29 WO disclosed
WO-2009130231-A1 PYRROLO [1, 2-A] PYRAZINE DERIVATIVES AS VASOPRESSIN VIB RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-10-29 WO disclosed