SCHEMBL4304424

SCHEMBL4304424

Fc1ccccc1[C@@H]1CO1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.48
KDM1B Q8NB78 1/20 0.48
TSHR P16473 2/20 0.46
HTR2C P28335 2/20 0.46
HTR2B P41595 2/20 0.46
CYP19A1 P11511 1/20 0.43
KDM4E B2RXH2 2/20 0.41
GAA P10253 2/20 0.41
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
ALDH1A1 P00352 2/20 0.38
RCOR1 Q9UKL0 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
NOS3 P29474 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29749063 1.00 KDM1A (0.48) KDM1AKDM1BTSHRHTR2CHTR2B
SCHEMBL30370466 1.00 KDM1A (0.48) KDM1AKDM1BTSHRHTR2CHTR2B
SCHEMBL937009 1.00 KDM1A (0.48) KDM1AKDM1BTSHRHTR2CHTR2B
SCHEMBL4753167 0.82 KDM1A (0.43) KDM1AKDM1BTSHRHTR2CHTR2B
SCHEMBL7055104 0.82 HTR2C (0.49) KDM1AKDM1BTSHRHTR2CHTR2B
SCHEMBL20833596 0.82 HTR2C (0.49) KDM1AKDM1BTSHRHTR2CHTR2B
SCHEMBL28759921 0.82 KDM1A (0.45) KDM1AKDM1BTSHRHTR2CHTR2B
SCHEMBL37732 0.82 TSHR (0.57) TSHRNOS3NOS2
SCHEMBL13224382 0.80 CHRNB2 (0.42) KDM1AKDM1BTSHRHTR2CHTR2B
SCHEMBL11358035 0.80 KDM1A (0.41) KDM1AKDM1BTSHRHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12540157-B2 Oxysterols and methods of use thereof Sage Therapeutics, LLC (US) 2026-02-03 US disclosed
US-12280023-B2 Fluorophenyl beta-hydroxyethylamines and their use in the treatment of hyperglycaemia ATROGI AB (SE) 2025-04-22 US disclosed
US-20240390298-A1 CYCLOHEXYL BETA-HYDROXY ALKYL AMINES AND MEDICAL USES THEREOF ATROGI AB (SE) 2024-11-28 US disclosed
EP-4405041-A1 CYCLOHEXYL BETA-HYDROXY ALKYL AMINES AND MEDICAL USES THEREOF Atrogi AB (SE) 2024-07-31 EP disclosed
US-20240199682-A1 OXYSTEROLS AND METHODS OF USE THEREOF SAGE THERAPEUTICS, INC. 2024-06-20 US disclosed
US-11851457-B2 Oxysterols and methods of use thereof SAGE THERAPEUTICS (US) 2023-12-26 US disclosed
US-20230364035-A1 FLUOROPHENYL BETA-HYDROXYETHYLAMINES AND THEIR USE IN THE TREATMENT OF HYPERGLYCAEMIA ATROGI AB (SE) 2023-11-16 US disclosed
EP-3681857-B1 FLUOROPHENYL BETA-HYDROXYETHYLAMINES AND THEIR USE IN THE TREATMENT OF HYPERGLYCAEMIA ATROGI AB (SE) 2023-11-08 EP disclosed
EP-4252848-A2 OXYSTEROLS AND METHODS OF USE THEREOF Sage Therapeutics, Inc. (US) 2023-10-04 EP disclosed
EP-4249054-A2 FLUOROPHENYL BETA-HYDROXYETHYLAMINES AND THEIR USE IN THE TREATMENT OF HYPERGLYCAEMIA Atrogi AB (SE) 2023-09-27 EP disclosed
US-4391826-A DIETETICS ELI LILLY AND COMPANY (US) 1983-07-05 US disclosed
EP-0007206-B1 PHENETHANOLAMINES, THEIR FORMULATIONS, PREPARATION AND USE ELI LILLY AND COMPANY (US) 1983-02-23 EP disclosed
EP-0006766-B1 PHENETHANOLAMINES, THEIR FORMULATIONS, USE AND PREPARATION ELI LILLY AND COMPANY (US) 1983-01-26 EP disclosed
EP-0007204-B1 PHENETHANOLAMINES, THEIR FORMULATIONS, USE AND PREPARATION ELI LILLY AND COMPANY (US) 1982-11-24 EP disclosed
EP-0048037-A1 Optically active 1-alkyl-3-(4-substituted-phenyl)-propylamines ELI LILLY AND COMPANY (US) 1982-03-24 EP disclosed
EP-0047536-A2 Substituted propylamines ELI LILLY AND COMPANY (US) 1982-03-17 EP disclosed
EP-0007206-A1 Phenethanolamines, their formulations, preparation and use ELI LILLY AND COMPANY (US) 1980-01-23 EP disclosed
EP-0007204-A1 Phenethanolamines, their formulations, use and preparation ELI LILLY AND COMPANY (US) 1980-01-23 EP disclosed
EP-0007205-A1 Optically active phenethanolamines, their formulations, use and preparation ELI LILLY AND COMPANY (US) 1980-01-23 EP disclosed
EP-0006766-A1 Phenethanolamines, their formulations, use and preparation ELI LILLY AND COMPANY (US) 1980-01-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240390298-A1 CYCLOHEXYL BETA-HYDROXY ALKYL AMINES AND MEDICAL USES THEREOF H1-5, CYP3A5, HRH3 KDM1A 1282/4885KDM1B 1425/4885TSHR 2693/4885
US-12540157-B2 Oxysterols and methods of use thereof HSD3B2, HSD3B1, HSD17B7 KDM1A 4209/4885KDM1B 4035/4885TSHR 1011/4885
US-20240199682-A1 OXYSTEROLS AND METHODS OF USE THEREOF NR1H3, NR1H2, HSD17B7 KDM1A 3351/4885KDM1B 3430/4885TSHR 998/4885
US-12280023-B2 Fluorophenyl beta-hydroxyethylamines and their use in the treatment of hyperglycaemia GPR119, SLC5A2, SLC5A1 KDM1A 1627/4885KDM1B 1528/4885TSHR 1556/4885
US-11851457-B2 Oxysterols and methods of use thereof NR1H3, NR1H2, HSD17B7 KDM1A 3233/4885KDM1B 3341/4885TSHR 915/4885
US-20230364035-A1 FLUOROPHENYL BETA-HYDROXYETHYLAMINES AND THEIR USE IN THE TREATMENT OF HYPERGLYCAEMIA GPR119, SLC5A2, SLC5A1 KDM1A 1627/4885KDM1B 1528/4885TSHR 1556/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.