SCHEMBL4306491

SCHEMBL4306491

NC(=O)CC=Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HB P07237 2/20 0.51
MEN1 O00255 1/20 0.51
LMNA P02545 1/20 0.51
HSP90AA1 P07900 1/20 0.51
MAPT P10636 1/20 0.51
PKM P14618 1/20 0.51
KMT2A Q03164 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
FBP1 P09467 1/20 0.50
RECQL P46063 1/20 0.50
MAOB P27338 5/20 0.49
NFE2L2 Q16236 1/20 0.49
HTT P42858 1/20 0.47
THRB P10828 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAOA P21397 1/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4321800 0.87 P4HB (0.48) P4HBMEN1LMNAHSP90AA1MAPT
SCHEMBL4989286 0.84 RECQL (0.52) P4HBMEN1LMNAHSP90AA1MAPT
SCHEMBL28669378 0.81 P4HB (0.48) P4HBMEN1LMNAHSP90AA1MAPT
SCHEMBL1124018 0.80 LMNA (0.62) P4HBMEN1LMNAHSP90AA1MAPT
SCHEMBL1124017 0.80 LMNA (0.62) P4HBMEN1LMNAHSP90AA1MAPT
SCHEMBL27279242 0.79 MAOB (0.48) P4HBMEN1LMNAHSP90AA1MAPT
SCHEMBL80957 0.79 NFE2L2 (0.56) P4HBMEN1LMNAHSP90AA1MAPT
SCHEMBL80956 0.79 NFE2L2 (0.56) P4HBMEN1LMNAHSP90AA1MAPT
SCHEMBL2095432 0.79 FBP1 (0.57) P4HBMEN1LMNAHSP90AA1MAPT
SCHEMBL2095430 0.79 FBP1 (0.57) P4HBMEN1LMNAHSP90AA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137338-A1 PYRAZOLE COMPOUNDS AS CCR1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-11-12 WO disclosed