SCHEMBL4306949

SCHEMBL4306949

CCCc1c(Cc2ccc(-c3ccccc3C#N)cc2)c(=O)nc(CC)n1-c1ccc(OC2(C(=O)O)CCCC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.40
PPARG P37231 2/20 0.37
FFAR1 O14842 1/20 0.37
AKR1B1 P15121 1/20 0.37
AGTR1 P30556 2/20 0.36
AGTR2 P50052 1/20 0.36
SLC33A1 O00400 3/20 0.35
GRIA2 P42262 1/20 0.34
GRIA4 P48058 1/20 0.34
ITGB1 P05556 1/20 0.34
ITGA4 P13612 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.33
APLNR P35414 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4319356 0.92 ACHE (0.38) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL1896768 0.82 ACHE (0.39) ACHEPPARGFFAR1AKR1B1SLC33A1
SCHEMBL1885478 0.82 ACHE (0.37) ACHEPPARGFFAR1AKR1B1SLC33A1
SCHEMBL4010015 0.81 PPARG (0.38) PPARGFFAR1AKR1B1AGTR1AGTR2
SCHEMBL4012069 0.80 SLC33A1 (0.43) PPARGFFAR1AKR1B1SLC33A1
SCHEMBL1890208 0.79 ACHE (0.42) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL13341905 0.78 ACHE (0.39) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL12349035 0.78 ACHE (0.40) ACHEPPARGFFAR1AKR1B1AGTR1
SCHEMBL13186066 0.77 ACHE (0.40) ACHEPPARGAGTR1SLC33A1APLNR
SCHEMBL4009738 0.76 AGTR1 (0.37) ACHEPPARGFFAR1AKR1B1AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed