SCHEMBL4010015

SCHEMBL4010015

CCCc1c(Cc2ccc(-c3ccccc3C#N)cc2)c(=O)nc(CC)n1-c1ccc(OC(C)(C)C(=O)OCC)cc1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.38
FFAR1 O14842 1/20 0.36
AKR1B1 P15121 1/20 0.36
AGTR1 P30556 1/20 0.35
AGTR2 P50052 1/20 0.35
PPARA Q07869 3/20 0.35
SLC33A1 O00400 2/20 0.34
ABCB11 O95342 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
HTR2A P28223 1/20 0.34
PMP22 Q01453 1/20 0.34
ALOX5AP P20292 1/20 0.34
PTPN1 P18031 1/20 0.34
APLNR P35414 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4017376 0.90 PPARA (0.38) PPARGFFAR1AKR1B1AGTR1AGTR2
SCHEMBL1890285 0.90 PPARG (0.38) PPARGFFAR1AKR1B1APLNR
SCHEMBL4011203 0.88 PPARG (0.36) PPARGFFAR1AKR1B1AGTR1AGTR2
SCHEMBL4009738 0.84 AGTR1 (0.37) PPARGFFAR1AKR1B1AGTR1AGTR2
SCHEMBL4319356 0.83 ACHE (0.38) PPARGFFAR1AKR1B1AGTR1AGTR2
SCHEMBL1892360 0.83
SCHEMBL4012069 0.83 SLC33A1 (0.43) PPARGFFAR1AKR1B1SLC33A1TSHR
SCHEMBL4306949 0.81 ACHE (0.40) PPARGFFAR1AKR1B1AGTR1AGTR2
SCHEMBL1892252 0.80 F10 (0.38) PPARGFFAR1AKR1B1AGTR1
SCHEMBL1893596 0.79 PPARG (0.41) PPARGFFAR1AKR1B1AGTR1APLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed