SCHEMBL4313643

SCHEMBL4313643

Oc1c(Cl)cc(-c2cnc(OCc3ccc(CNCCc4ccccc4N4CCOCC4)cc3)nn2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.40
SCN2A Q99250 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
P2RX7 Q99572 1/20 0.35
HDAC1 Q13547 2/20 0.35
KDM1A O60341 1/20 0.35
DYRK1A Q13627 1/20 0.35
WDR5 P61964 1/20 0.34
GAA P10253 3/20 0.34
LMNA P02545 1/20 0.34
MCOLN3 Q8TDD5 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313635 0.79 DYRK1A (0.38) HDAC1KDM1ADYRK1AGAALMNA
SCHEMBL8017379 0.78 MELK (0.43) CHEK1MEN1KMT2ADYRK1ANPC1
SCHEMBL3240064 0.76 ROCK2 (0.39) MEN1KMT2ADYRK1AGAAALDH1A1
SCHEMBL3242799 0.75 SMN1; SMN2 (0.44) MEN1KMT2AHDAC1LMNAALDH1A1
SCHEMBL3241352 0.74 MAPK1 (0.43) MEN1KMT2A
SCHEMBL3237578 0.73 DRD2 (0.45) KMT2ALMNANPC1ALDH1A1MAPT
SCHEMBL3236041 0.73 SMN1; SMN2 (0.40) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3239905 0.73 SMN1; SMN2 (0.45) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3244194 0.72 DRD4 (0.46) MEN1KMT2APOLB
SCHEMBL3243794 0.72 ENPP2 (0.40) LMNANPC1ALDH1A1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009131958-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING TRIAZINE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO claimed