SCHEMBL4313635

SCHEMBL4313635

CCN(Cc1ccc(COc2ncc(-c3cc(Cl)c(O)c(Cl)c3)nn2)cc1)c1ccccc1N1CCOCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.38
HCAR1 Q9BXC0 4/20 0.33
PDK1 Q15118 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
CNR2 P34972 2/20 0.33
CNR1 P21554 1/20 0.33
GAA P10253 2/20 0.32
LMNA P02545 2/20 0.32
MCOLN3 Q8TDD5 1/20 0.32
CYP11B2 P19099 1/20 0.32
PDE10A Q9Y233 1/20 0.32
KDM1A O60341 1/20 0.32
HDAC1 Q13547 1/20 0.32
BCHE P06276 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
CCR5 P51681 1/20 0.32
PIK3CA P42336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313643 0.79 CHEK1 (0.40) DYRK1ACNR2CNR1GAALMNA
SCHEMBL8017379 0.78 MELK (0.43) DYRK1ANPC1RAB9ACCR5L3MBTL1
SCHEMBL3240022 0.77 L3MBTL1 (0.46) DYRK1ABCHEALDH1A1MAPK1L3MBTL1
SCHEMBL3232831 0.77 OPRK1 (0.40) GAAALDH1A1MAPK1
SCHEMBL3240305 0.76 PDK1 (0.41) PDK1BCHENPC1RAB9AL3MBTL1
SCHEMBL3245515 0.75 CCR5 (0.42) DYRK1AGAABCHEMAPTCCR5
SCHEMBL3241365 0.75 ACHE (0.45) PDK1CNR2CNR1KDM1AHDAC1
SCHEMBL3238195 0.74 L3MBTL1 (0.36) DYRK1AGAALMNABCHEALDH1A1
SCHEMBL3240064 0.74 ROCK2 (0.39) DYRK1AGAAALDH1A1MAPK1
SCHEMBL3237578 0.73 DRD2 (0.45) LMNAALDH1A1MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009131958-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING TRIAZINE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO claimed