SCHEMBL3240064

SCHEMBL3240064

Oc1c(Cl)cc(-c2cnc(OCc3ccc(CNC(CN4CCOCC4)c4ccccc4)cc3)nn2)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
HSD17B13 Q7Z5P4 1/20 0.37
KMT2A Q03164 2/20 0.37
GAA P10253 1/20 0.37
MAPK1 P28482 3/20 0.37
GPR88 Q9GZN0 1/20 0.36
CTSS P25774 1/20 0.36
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
SCN1A P35498 2/20 0.35
SCN5A Q14524 2/20 0.35
SCN8A Q9UQD0 2/20 0.35
NOX1 Q9Y5S8 1/20 0.35
MAP3K8 P41279 1/20 0.35
PDE5A O76074 1/20 0.35
ERBB2 P04626 2/20 0.34
DYRK1A Q13627 1/20 0.34
MELK Q14680 1/20 0.34
EGFR P00533 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3240063 0.93 ROCK2 (0.37) ROCK2ROCK1KMT2AMAPK1GPR88
SCHEMBL3243937 0.92 GPR88 (0.39) ROCK2ROCK1HSD17B13KMT2AGAA
SCHEMBL3237511 0.91 ROCK2 (0.38) ROCK2ROCK1KMT2AGAAMAPK1
SCHEMBL3232831 0.86 OPRK1 (0.40) ROCK2ROCK1HSD17B13KMT2AGAA
SCHEMBL8017379 0.83 MELK (0.43) KMT2AMEN1DYRK1AMELK
SCHEMBL3239887 0.81 MEN1 (0.36) KMT2AMAPK1MEN1DYRK1A
SCHEMBL3240305 0.76 PDK1 (0.41) KMT2AMEN1MELK
SCHEMBL3237578 0.76 DRD2 (0.45) KMT2AALDH1A1
SCHEMBL4313643 0.76 CHEK1 (0.40) KMT2AGAAALDH1A1MEN1DYRK1A
SCHEMBL3241365 0.75 ACHE (0.45) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090264433-A1 Compounds, Compositions and Methods Comprising Triazine Derivatives INSTITUTE FOR ONEWORLD HEALTH 2009-10-22 US claimed
US-20100144733-A1 Compounds, compositions and methods comprising heteroaromatic derivatives INSTITUTE FOR ONEWORLD HEALTH 2010-06-10 US disclosed
US-20100144733-A1 Compounds, compositions and methods comprising heteroaromatic derivatives INSTITUTE FOR ONEWORLD HEALTH 2010-06-10 US disclosed
US-20100144733-A1 Compounds, compositions and methods comprising heteroaromatic derivatives INSTITUTE FOR ONEWORLD HEALTH 2010-06-10 US disclosed
US-20090318429-A1 Compounds, Compositions and Methods Comprising Heteroaromatic Derivatives INSTITUTE FOR ONEWORLD HEALTH 2009-12-24 US disclosed
US-20090318429-A1 Compounds, Compositions and Methods Comprising Heteroaromatic Derivatives INSTITUTE FOR ONEWORLD HEALTH 2009-12-24 US disclosed
US-20090318429-A1 Compounds, Compositions and Methods Comprising Heteroaromatic Derivatives INSTITUTE FOR ONEWORLD HEALTH 2009-12-24 US disclosed
US-20090264433-A1 Compounds, Compositions and Methods Comprising Triazine Derivatives INSTITUTE FOR ONEWORLD HEALTH 2009-10-22 US disclosed
US-20090264433-A1 Compounds, Compositions and Methods Comprising Triazine Derivatives INSTITUTE FOR ONEWORLD HEALTH 2009-10-22 US disclosed
US-20090264433-A1 Compounds, Compositions and Methods Comprising Triazine Derivatives INSTITUTE FOR ONEWORLD HEALTH 2009-10-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090264433-A1 Compounds, Compositions and Methods Comprising Triazine Derivatives CFTR, PKD1, PKD2 ROCK2 2675/4885ROCK1 2390/4885HSD17B13 2679/4885
US-20100144733-A1 Compounds, compositions and methods comprising heteroaromatic derivatives CFTR, PKD1, PKD2 ROCK2 3358/4885ROCK1 2801/4885HSD17B13 924/4885
US-20090318429-A1 Compounds, Compositions and Methods Comprising Heteroaromatic Derivatives CFTR, PKD1, PKD2 ROCK2 3358/4885ROCK1 2801/4885HSD17B13 924/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.