SCHEMBL4316682

SCHEMBL4316682

COC(=O)c1cc(OC)ccc1C#N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56
CYP3A4 P08684 1/20 0.56
KDM4E B2RXH2 4/20 0.55
GAA P10253 2/20 0.50
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
HSD17B10 Q99714 3/20 0.49
TP53 P04637 2/20 0.49
NR4A2 P43354 1/20 0.48
HPGD P15428 1/20 0.47
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
ALDH1A1 P00352 2/20 0.44
GLA P06280 2/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17197313 0.87 CYP1A2 (0.56) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL4309752 0.85 SMN1; SMN2 (0.54) KDM4ENPC1RAB9AHSD17B10TP53
SCHEMBL25256914 0.85 CA12 (0.61) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL7369021 0.84 KDM4E (0.52) CYP1A2CYP2C9CYP2C19CYP3A4KDM4E
SCHEMBL23716298 0.84 CYP1A2 (0.45) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL30744989 0.84 HPGD (0.46) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL27145832 0.84 ACACB (0.47) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL8324473 0.83 NPC1 (0.47) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL8324669 0.83 PARP1 (0.49) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL5846153 0.81 GAA (0.51) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106188029-B Two and ring class anaplastic lymphoma kinase inhibitor 山东轩竹医药科技有限公司 2018-09-18 CN disclosed
US-20090258885-A1 Diphenylmethane Derivatives as Inhibitors of Leukotriene Biosynthesis MERCK SHARP & DOHME CORP. 2009-10-15 US disclosed
US-20090258885-A1 Diphenylmethane Derivatives as Inhibitors of Leukotriene Biosynthesis MERCK SHARP & DOHME CORP. 2009-10-15 US disclosed
US-20090258885-A1 Diphenylmethane Derivatives as Inhibitors of Leukotriene Biosynthesis MERCK SHARP & DOHME CORP. 2009-10-15 US disclosed
WO-2008020306-A2 ISOINDOLE DERIVATIVES PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed
WO-2008020306-A2 ISOINDOLE DERIVATIVES PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090258885-A1 Diphenylmethane Derivatives as Inhibitors of Leukotriene Biosynthesis LTC4S, LTA4H, ALOX5 CYP1A2 670/4885CYP2D6 756/4885CYP2C9 1708/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.