SCHEMBL4324285

SCHEMBL4324285

CN(C)c1cccc2c(S(=O)(=O)Oc3ccc(-c4csc(N=C(N)N)n4)cc3)cccc12

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 16/20 0.52
ATP4B P51164 16/20 0.52
NPC1 O15118 2/20 0.52
MAPT P10636 2/20 0.52
RAB9A P51151 2/20 0.52
GFER P55789 1/20 0.47
F2 P00734 3/20 0.45
PRSS1 P07477 3/20 0.45
PRSS2 P07478 3/20 0.45
PRSS3 P35030 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4324290 0.82 HSPA5 (0.52) NPC1MAPTRAB9AF2PRSS1
SCHEMBL4324082 0.75 ATP4A (0.64) ATP4AATP4BNPC1MAPTRAB9A
SCHEMBL4330186 0.75 MAPT (0.69) ATP4AATP4BNPC1MAPTRAB9A
SCHEMBL4334951 0.75 ATP4A (0.58) ATP4AATP4BNPC1MAPTRAB9A
SCHEMBL711797 0.71 CA2 (0.58) F2PRSS1PRSS2PRSS3
SCHEMBL4322753 0.71 ATP4A (0.55) ATP4AATP4BNPC1MAPTRAB9A
SCHEMBL16610066 0.71 TYMS (0.53) F2PRSS1PRSS2PRSS3
SCHEMBL4109611 0.70 ATP4A (1.00) ATP4AATP4BNPC1MAPTRAB9A
SCHEMBL4322564 0.70 ATP4A (0.54) ATP4AATP4BNPC1MAPTRAB9A
SCHEMBL4342349 0.69 ATP4A (0.56) ATP4AATP4BNPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO claimed
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO disclosed