Clorindione

Clorindione

SCHEMBL43305

O=C1c2ccccc2C(=O)C1c1ccc(Cl)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 1.00
MAPT P10636 5/20 0.68
TP53 P04637 3/20 0.68
LMNA P02545 2/20 0.68
MAPK1 P28482 2/20 0.68
CYP1A2 P05177 1/20 0.68
CYP3A4 P08684 1/20 0.68
HTR2B P41595 1/20 0.68
MEN1 O00255 5/20 0.64
KMT2A Q03164 5/20 0.64
NPC1 O15118 5/20 0.64
KDM4E B2RXH2 2/20 0.64
GAA P10253 2/20 0.64
SMN1; SMN2 Q16637 3/20 0.59
MAPK10 P53779 1/20 0.59
HPGD P15428 1/20 0.58
MAOA P21397 1/20 0.58
PTGS2 P35354 1/20 0.58
GSK3B P49841 1/20 0.51
ALDH1A1 P00352 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenindione SCHEMBL29388073 0.81 MAPT (1.00) RAB9AMAPTTP53LMNAMAPK1
Phenindione SCHEMBL33831 0.81 MAPT (1.00) RAB9AMAPTTP53LMNAMAPK1
SCHEMBL10620936 0.81 RAB9A (0.67) RAB9AMAPTTP53LMNAMAPK1
SCHEMBL14939892 0.80 RAB9A (0.67) RAB9AMAPTTP53LMNAMAPK1
SCHEMBL17525348 0.80 MAPT (0.71) RAB9AMAPTTP53LMNAMAPK1
SCHEMBL10620960 0.80 RAB9A (0.66) RAB9AMAPTTP53LMNAMAPK1
Phenindione SCHEMBL1443973 0.79 MAPT (0.95) RAB9AMAPTTP53LMNAMAPK1
Phenindione SCHEMBL6827577 0.79 MAPT (0.95) RAB9AMAPTTP53LMNAMAPK1
SCHEMBL10559114 0.79 MAPT (0.95) RAB9AMAPTTP53LMNAMAPK1
SCHEMBL5649473 0.78 KMT2A (1.00) RAB9AMAPTTP53LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1591 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11421234-B2 Aptamers for targeting coagulation factor XIII and uses thereof CHANG GUNG UNIVERSITY (TW) 2022-08-23 US claimed
EP-3964208-A1 COMPOSITION COMPRISING ISOQUERCETIN FOR TREATING VENOUS THROMBOSIS Quercegen Pharmaceuticals LLC (US) 2022-03-09 EP claimed
US-20210371512-A1 Use of IL-1 beta Binding Antibodies NOVARTIS AG (CH) 2021-12-02 US claimed
US-20210163945-A1 APTAMERS FOR TARGETING COAGULATION FACTOR XIII AND USES THEREOF CHANG GUNG UNIVERSITY (TW) 2021-06-03 US claimed
WO-2021054927-A2 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS SOUTH DAKOTA BOARD OF REGENTS (US) 2021-03-25 WO claimed
US-20200147264-A1 DETECTION OF BIOPROSTHETIC VALVE DEGENERATION ASSISTANCE PUBLIQUE-HOPITAUX DE PARIS (FR) 2020-05-14 US claimed
US-20200048305-A1 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS SOUTH DAKOTA BOARD OF REGENTS (US) 2020-02-13 US claimed
EP-3100728-B1 PHARMACEUTICAL COMPOSITIONS COMPRISING PRASUGREL AND CYCLODEXTRIN DERIVATIVES AND METHODS OF MAKING AND USING THE SAME CYDEX PHARMACEUTICALS INC (US) 2019-11-20 EP claimed
US-10391096-B2 Method for treating thrombotic disorders using quercetin-containing compositions QUERCEGEN PHARMACEUTICALS LLC (US) 2019-08-27 US claimed
US-20180177759-A1 COMBINATION OF AN ANTIANDROGEN WITH A VITAMIN K ANTAGONIST OR WITH A GAMMA-GLUTAMYL CARBOXYLASE INHIBITOR FOR THE THERAPY OF ANDROGEN RECEPTOR POSITIVE CANCER CEMM - FORSCHUNGSZENTRUM FÜR MOLEKULARE MEDIZIN GMBH (AT) 2018-06-28 US claimed
US-20020173818-A1 Delivering an agent to a patient's body BOSTON SCIENTIFIC SCIMED, INC. 2002-11-21 US claimed
WO-2002091957-A1 DELIVERING AN AGENT TO A PATIENT'S BODY SCIMED LIFE SYSTEM, INC. (US) 2002-11-21 WO claimed
WO-2002049649-A2 PHARMACEUTICAL FORMULATION CONTAINING THIENOPYRIMIDINES AND ANTITHROMBOTICS, CALCIUM ANTAGONISTS, PROSTAGLANDINS OR PROSTAGLANDIN DERIVATIVES (2) MERCK PATENT GMBH (DE) 2002-06-27 WO claimed
WO-2002049650-A2 PHARMACEUTICAL FORMULATION CONTAINING THIENOPYRIMIDINES AND ANTITHROMBOTICS, CALCIUM ANTAGONISTS, PROSTAGLANDINS OR PROSTAGLANDIN DERIVATIVES MERCK PATENT GMBH (DE) 2002-06-27 WO claimed
WO-2002049651-A1 PHARMACEUTICAL FORMULATION CONTAINING PYRAZOLO[4,3-D]PYRIMIDINES AND ANTITHROMBOTIC AGENTS, CALCIUM-ANTAGONISTS, PROSTAGLANDINS OR PROSTAGLANDIN DERIVATIVES MERCK PATENT GMBH (DE) 2002-06-27 WO claimed
EP-1100479-A1 MEDICINAL PRODUCTS WITH RETARDED PHARMACOLOGICAL ACTIVITY AND METHOD FOR THE PRODUCTION THEREOF Schierholz, Jörg, Dr.Dr. (DE) 2001-05-23 EP claimed
EP-0985413-A1 Medical articles with sustained pharmacological activity and process for their preparation Schierholz, Jörg Michael, Dr. Dr. (DE) 2000-03-15 EP claimed
WO-2000007574-A1 MEDICINAL PRODUCTS WITH RETARDED PHARMACOLOGICAL ACTIVITY AND METHOD FOR THE PRODUCTION THEREOF SCHIERHOLZ JOERG (DE) 2000-02-17 WO claimed
EP-0088051-B1 RODENTICIDAL BAIT CIBA-GEIGY AG (CH) 1986-11-12 EP claimed
EP-0088051-A1 Rodenticidal bait CIBA-GEIGY AG (CH) 1983-09-07 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200048305-A1 GLUTATHIONE-CHOLESTEROL DERIVATIVES AS BRAIN TARGETING AGENTS GSTK1, GSTO1, GSTM2 RAB9A 1626/4885MAPT 1050/4885TP53 4095/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.