SCHEMBL4331865

SCHEMBL4331865

COc1ccc(-c2ccc(C(=O)Oc3ccc(-c4csc(N=C(N)N)n4)cc3)cc2)cc1

nearest known ligand 0.76

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 14/20 0.76
ATP4B P51164 14/20 0.76
NPC1 O15118 3/20 0.76
RAB9A P51151 3/20 0.76
MAPT P10636 2/20 0.76
ACR P10323 2/20 0.57
PRSS1 P07477 1/20 0.57
GFER P55789 1/20 0.55
MEN1 O00255 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CSNK2A1 P68400 1/20 0.48
HGFAC Q04756 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4322678 0.91 ATP4A (0.70) ATP4AATP4BNPC1RAB9AMAPT
SCHEMBL4329794 0.90 ATP4A (0.66) ATP4AATP4BNPC1RAB9AMAPT
SCHEMBL4330723 0.87 PRSS1 (0.61) ATP4AATP4BNPC1RAB9AMAPT
SCHEMBL4109611 0.87 ATP4A (1.00) ATP4AATP4BNPC1RAB9AMAPT
Bromide SCHEMBL826017 0.86 ATP4A (1.00) ATP4AATP4BNPC1RAB9AMAPT
SCHEMBL4324204 0.84 ATP4A (0.55) ATP4AATP4BNPC1RAB9AMAPT
SCHEMBL4333457 0.83 ATP4A (0.57) ATP4AATP4BNPC1RAB9AMAPT
SCHEMBL4326705 0.83 ATP4A (0.55) ATP4AATP4BNPC1RAB9AMAPT
SCHEMBL4331871 0.78 ADORA3 (0.58) NPC1RAB9AMAPTMEN1KDM4E
SCHEMBL4342349 0.76 ATP4A (0.56) ATP4AATP4BNPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO claimed
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO disclosed