SCHEMBL4331871

SCHEMBL4331871

COc1ccc(-c2ccc(C(=O)Oc3ccc(-c4csc(NC(=N)N)n4)cc3)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.58
CSNK2A1 P68400 1/20 0.57
GSTO1 P78417 1/20 0.56
RAB9A P51151 7/20 0.56
KDM4E B2RXH2 2/20 0.56
SMN1; SMN2 Q16637 4/20 0.55
LMNA P02545 4/20 0.55
MAPK1 P28482 5/20 0.55
ALDH1A1 P00352 5/20 0.55
NPSR1 Q6W5P4 2/20 0.55
RXFP1 Q9HBX9 1/20 0.55
MEN1 O00255 6/20 0.54
KMT2A Q03164 6/20 0.54
NPC1 O15118 5/20 0.54
MAPT P10636 5/20 0.54
TP53 P04637 2/20 0.54
PTGS2 P35354 1/20 0.52
GAA P10253 1/20 0.51
ROCK1 Q13464 2/20 0.51
RECQL P46063 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4322683 0.91 MEN1 (0.60) ADORA3CSNK2A1GSTO1RAB9AKDM4E
SCHEMBL4329797 0.90 ADORA3 (0.56) ADORA3CSNK2A1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL3595657 0.88 PTGS2 (0.66) ADORA3CSNK2A1GSTO1RAB9ASMN1; SMN2
SCHEMBL4330728 0.88 ADORA3 (0.48) ADORA3CSNK2A1GSTO1RAB9AKDM4E
SCHEMBL3615150 0.86 MEN1 (0.55) ADORA3CSNK2A1GSTO1RAB9AKDM4E
SCHEMBL4324209 0.85 RAB9A (0.44) ADORA3CSNK2A1GSTO1RAB9AKDM4E
SCHEMBL4333461 0.84 RAB9A (0.53) ADORA3CSNK2A1GSTO1RAB9AKDM4E
SCHEMBL4326708 0.84 MAPT (0.53) ADORA3RAB9ASMN1; SMN2LMNAMAPK1
SCHEMBL3601789 0.83 KDM4E (0.60) ADORA3GSTO1RAB9AKDM4ESMN1; SMN2
SCHEMBL13578642 0.81 MAPK1 (0.44) ADORA3CSNK2A1GSTO1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO claimed
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO disclosed
WO-2009146013-A1 MYOSIN LIGHT CHAIN PHOSPHATASE INHIBITORS GEORGETOWN UNIVERSITY (US) 2009-12-03 WO disclosed