SCHEMBL43350

SCHEMBL43350

O=C(O)C(Cc1ccccc1)NCP(=O)(O)O

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MME P08473 4/20 0.62
ECE1 P42892 3/20 0.62
MEN1 O00255 1/20 0.62
KMT2A Q03164 1/20 0.62
LAP3 P28838 3/20 0.54
ANPEP P15144 1/20 0.54
ACE P12821 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL43351 1.00 MME (0.62) MMEECE1MEN1KMT2ALAP3
SCHEMBL7411127 0.92 MME (0.62) MMEECE1MEN1KMT2AACE
SCHEMBL7411123 0.92 MME (0.62) MMEECE1MEN1KMT2AACE
SCHEMBL3098759 0.87 LAP3 (0.56) MMEECE1MEN1KMT2ALAP3
SCHEMBL3098754 0.87 LAP3 (0.56) MMEECE1MEN1KMT2ALAP3
SCHEMBL2989598 0.87 MME (0.56) MMEECE1MEN1KMT2AACE
SCHEMBL2996598 0.87 MME (0.56) MMEECE1MEN1KMT2AACE
SCHEMBL16415834 0.86 MME (0.49) MMEECE1MEN1KMT2AL3MBTL1
SCHEMBL7311905 0.85 MME (0.73) MMEECE1ACE
SCHEMBL2995625 0.84 ANPEP (0.53) MMEECE1MEN1KMT2AANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1109 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230364178-A1 Small Molecule Cancer Treatments that Cause Necrosis in Cancer Cells But Do Not Affect Normal Cells UNIV NEW YORK STATE RES FOUND (US) 2023-11-16 US claimed
US-20210205403-A1 Small Molecule Cancer Treatments that Cause Necrosis in Cancer Cells But Do Not Affect Normal Cells THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK 2021-07-08 US claimed
US-20200038471-A1 SMALL MOLECULE CANCER TREATMENTS THAT CAUSE NECROSIS IN CANCER CELLS BUT DO NOT AFFECT NORMAL CELLS THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK 2020-02-06 US claimed
US-20170209521-A1 SMALL MOLECULE CANCER TREATMENTS THAT CAUSE NECROSIS IN CANCER CELLS BUT DO NOT AFFECT NORMAL CELLS THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK 2017-07-27 US claimed
US-20110183915-A1 Small Molecule Cancer Treatments that cause Necrosis in Cancer Cells but do not Affect Normal Cells THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK 2011-07-28 US claimed
US-20110034670-A1 BISUBSTRATE INHIBITORS OF PROTEIN KINASES AS THERAPEUTIC AGENTS BOARD OF GOVERNORS FOR HIGHER EDUCATION, STATE OF RHODE ISLAND AND PROVIDENCE PLANTATIONS (US) 2011-02-10 US claimed
US-7871981-B2 Inhibition of cell motility, angiogenesis, and metastasis THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-01-18 US claimed
EP-2224961-A1 SMALL MOLECULE CANCER TREATMENTS THAT CAUSE NECROSIS IN CANCER CELLS BUT DO NOT AFFECT NORMAL CELLS The Research Foundation of the State University of New York (US) 2010-09-08 EP claimed
US-7776844-B2 N-(phosphonoalkyl)-amino acids, derivatives thereof and compositions and methods of use YU RUEY J 2010-08-17 US claimed
US-20090208499-A1 N-(Phosphonoalkyl)-Amino Acids, Derivatives Thereof and Compositions and Methods of Use YU RUEY J 2009-08-20 US claimed
US-5801149-A PEPTIDS FOR INHIBITION OF PROTEINS JOSLIN D-ABETES CENTER, INC. (US) 1998-09-01 US claimed
EP-0846127-A1 ACYLATED OLIGOPEPTIDE DERIVATIVES HAVING CELL SIGNAL INHIBITING ACTIVITY Novartis AG (CH) 1998-06-10 EP claimed
EP-0845217-A1 Inhibiting undesirable taste in oral compositions THE PROCTER & GAMBLE COMPANY (US) 1998-06-03 EP claimed
EP-0768821-A1 pp60PIK : A DOWNSTREAM ELEMENT IN INSULIN SIGNALING THE JOSLIN DIABETES CENTER, INC. (US) 1997-04-23 EP claimed
WO-1997008193-A1 ACYLATED OLIGOPEPTIDE DERIVATIVES HAVING CELL SIGNAL INHIBITING ACTIVITY NOVARTIS AG (CH) 1997-03-06 WO claimed
WO-1997007131-A1 ACYLATED OLIGOPEPTIDES CONTAINING PHOSPHOTYROSINE AS INHIBITORS OF PROTEIN TYROSINE KINASES NOVARTIS AG (CH) 1997-02-27 WO claimed
WO-1996032411-A1 BINDING SITES FOR PHOSPHOTYROSINE BINDING DOMAINS KAVANAUGH WILLIAM MICHAEL (US) 1996-10-17 WO claimed
WO-1995034201-A1 pp60PIK: A DOWNSTREAM ELEMENT IN INSULIN SIGNALING JOSLIN DIABETES CENTER, INC. (US) 1995-12-21 WO claimed
WO-1994008600-A1 INHIBITION OF SIGNAL TRANSDUCTION MOLECULES JOSLIN DIABETES CENTER (US) 1994-04-28 WO claimed
WO-1994007913-A1 PEPTIDE ANTAGONISTS OF SH2 BINDING AND THERAPEUTIC USES THEREOF WARNER-LAMBERT COMPANY (US) 1994-04-14 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110183915-A1 Small Molecule Cancer Treatments that cause Necrosis in Cancer Cells but do not Affect Normal Cells HMGB2, HMGB1, HMGB3 MME 384/4885ECE1 2587/4885MEN1 715/4885
US-20200038471-A1 SMALL MOLECULE CANCER TREATMENTS THAT CAUSE NECROSIS IN CANCER CELLS BUT DO NOT AFFECT NORMAL CELLS HMGB2, HMGB1, HMGB3 MME 384/4885ECE1 2587/4885MEN1 715/4885
US-20170209521-A1 SMALL MOLECULE CANCER TREATMENTS THAT CAUSE NECROSIS IN CANCER CELLS BUT DO NOT AFFECT NORMAL CELLS HMGB2, HMGB1, HMGB3 MME 384/4885ECE1 2587/4885MEN1 715/4885
US-20110034670-A1 BISUBSTRATE INHIBITORS OF PROTEIN KINASES AS THERAPEUTIC AGENTS SRC, PDXK, DSTYK MME 845/4885ECE1 3196/4885MEN1 3316/4885
US-20210205403-A1 Small Molecule Cancer Treatments that Cause Necrosis in Cancer Cells But Do Not Affect Normal Cells HMGB2, HMGB1, HMGB3 MME 384/4885ECE1 2587/4885MEN1 715/4885
US-20230364178-A1 Small Molecule Cancer Treatments that Cause Necrosis in Cancer Cells But Do Not Affect Normal Cells HMGB2, HMGB1, HMGB3 MME 384/4885ECE1 2587/4885MEN1 715/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.