SCHEMBL433543

SCHEMBL433543

Fc1cc(Cl)ccc1-c1c(Cl)[c]ccc1F

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.36
KMO O15229 2/20 0.35
EGLN2 Q96KS0 1/20 0.34
GRM2 Q14416 3/20 0.33
HSD11B1 P28845 1/20 0.32
FASN P49327 1/20 0.32
S100A4 P26447 1/20 0.31
PDE4A P27815 2/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
MAPK14 Q16539 1/20 0.30
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
TP53 P04637 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
PDK2 Q15119 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17514805 0.88 GRM2 (0.35) PTGS2KMOEGLN2GRM2HSD11B1
SCHEMBL434637 0.88 AHR (0.39) HSD11B1MAPK14KDM4ENPC1TP53
SCHEMBL432660 0.86 ALDH1A1 (0.34) PTGS2KMOGRM2MAPK14KDM4E
SCHEMBL433574 0.86 KMO (0.35) PTGS2KMOEGLN2GRM2HSD11B1
SCHEMBL17514628 0.83 PTGS2 (0.34) PTGS2KMOEGLN2GRM2HSD11B1
SCHEMBL17514857 0.83 PTGS2 (0.37) PTGS2KMOEGLN2GRM2HSD11B1
SCHEMBL1274798 0.82 HSD11B1 (0.42) PTGS2KMOEGLN2GRM2HSD11B1
SCHEMBL17514578 0.79 KMO (0.40) PTGS2KMOEGLN2GRM2HSD11B1
SCHEMBL432908 0.78 PTGS1 (0.34) HSD11B1KDM4ENPC1RAB9APDK2
SCHEMBL17514653 0.77 NISCH (0.37) GRM2HSD11B1FASNMAPK14KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7151097-B2 Bicyclic pyrazolyl and imidazolyl compounds and uses thereof PFIZER INC. (US) 2006-12-19 US claimed
WO-2016026830-A1 NOVEL FUNGICIDAL PYRAZOLE DERIVATIVES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-02-25 WO disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
EP-0121979-B1 AZOLYLMETHYL TETRAHYDROFURAN DERIVATIVES AS PLANT GROWTH REGULATORS AND FUNGICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-09-26 EP disclosed