SCHEMBL4336046

SCHEMBL4336046

CC(C)(C)c1ccc(C(=O)NCCCCn2cc(-c3ccccc3)c3ccc(C(=O)O)cc32)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
GAA P10253 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 4/20 0.45
NPC1 O15118 2/20 0.45
NR1H4 Q96RI1 3/20 0.44
TMEM97 Q5BJF2 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
SCN9A Q15858 1/20 0.43
POLB P06746 1/20 0.43
CASP3 P42574 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
ESRRG P62508 1/20 0.42
EPHX2 P34913 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4324148 0.90 SCN9A (0.46) MAPTTMEM97SIGMAR1SCN9A
SCHEMBL4320012 0.90 LMNA (0.46) LMNAALDH1A1RAB9ANPC1TMEM97
SCHEMBL4333849 0.88 DRD2 (0.46) MAPTSMN1; SMN2TMEM97SIGMAR1DRD2
SCHEMBL4325414 0.88 KMT2A (0.47) DRD2DRD3SCN9AKMT2A
SCHEMBL4330789 0.88 NPC1 (0.49) LMNASMN1; SMN2RAB9ANPC1DRD2
SCHEMBL4331873 0.88 NPC1 (0.50) ALDH1A1MAPTSMN1; SMN2HTTRAB9A
SCHEMBL4326354 0.85 NAMPT (0.46) NR1H4DRD2DRD3SCN9AEPHX2
SCHEMBL4324654 0.84 NPC1 (0.46) RAB9ANPC1SCN9A
SCHEMBL4321416 0.84 DRD2 (0.46) LMNAALDH1A1MAPTSMN1; SMN2GAA
SCHEMBL4326720 0.83 DRD3 (0.47) LMNARAB9ANPC1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO disclosed