SCHEMBL433724

SCHEMBL433724

Cc1cn2cc(Cl)ccc2n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 10/20 0.56
NPC1 O15118 7/20 0.56
KDM4E B2RXH2 8/20 0.54
TP53 P04637 1/20 0.54
MAPT P10636 5/20 0.54
SMN1; SMN2 Q16637 5/20 0.53
ALDH1A1 P00352 5/20 0.53
POLB P06746 3/20 0.53
LMNA P02545 1/20 0.53
CASP3 P42574 1/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53
SENP6 Q9GZR1 1/20 0.53
APP P05067 1/20 0.50
HRH4 Q9H3N8 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4790793 0.80 NPC1 (0.59) RAB9ANPC1KDM4ETP53MAPT
SCHEMBL7911725 0.78 RAB9A (0.60) RAB9ANPC1KDM4ETP53MAPT
SCHEMBL1664803 0.76 RAB9A (0.83) RAB9ANPC1KDM4ETP53MAPT
SCHEMBL3486359 0.75 PIK3CG (0.60) RAB9ANPC1KDM4ETP53MAPT
SCHEMBL19086855 0.75 RAB9A (0.56) RAB9ANPC1KDM4ETP53MAPT
SCHEMBL12778714 0.75 RAB9A (0.56) RAB9ANPC1KDM4ETP53MAPT
SCHEMBL7988504 0.75 APP (0.50) RAB9ANPC1KDM4ETP53MAPT
SCHEMBL14427902 0.75 CYP11B1 (0.57) RAB9ANPC1KDM4ETP53SMN1; SMN2
SCHEMBL13391848 0.75 APP (0.42) RAB9ANPC1KDM4ETP53MAPT
SCHEMBL2294229 0.75 APP (0.50) RAB9ANPC1KDM4ETP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 57 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230312481-A1 SUBSTITUTED (PHTHALAZIN-1-YLMETHYL)UREAS, SUBSTITUTED N-(PHTHALAZIN-1-YLMETHYL)AMIDES, AND ANALOGUES THEREOF ARBUTUS BIOPHARMA CORP (CA) 2023-10-05 US disclosed
US-20230312481-A1 SUBSTITUTED (PHTHALAZIN-1-YLMETHYL)UREAS, SUBSTITUTED N-(PHTHALAZIN-1-YLMETHYL)AMIDES, AND ANALOGUES THEREOF ARBUTUS BIOPHARMA CORP (CA) 2023-10-05 US disclosed
US-11168083-B2 Inhibitors of Plasma Kallikrein and uses thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-11-09 US disclosed
US-11136310-B2 Iminotetrahydropyrimidinone derivatives as plasmepsin V inhibitors UCB Biopharma SRL (BE) 2021-10-05 US disclosed
US-11112366-B2 Reagent and kit for enhancing chemiluminescent reaction NATIONAL TAIWAN OCEAN UNIVERSITY (TW) 2021-09-07 US disclosed
CN-108290860-B Iminotetrahydropyrimidinone derivatives as PLASMEPSIN V inhibitors UCB生物制药有限责任公司 2021-08-10 CN disclosed
WO-2021126729-A1 PRMT5 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2021-06-24 WO disclosed
EP-3438095-B1 PYRIDAZINONE COMPOUND OR ITS SALT, AND HERBICIDE CONTAINING IT ISHIHARA SANGYO KAISHA (JP) 2021-06-16 EP disclosed
US-10870638-B2 Pyridazinone compound or its salt, and herbicide containing it ISHIHARA SANGYO KAISHA, LTD. (JP) 2020-12-22 US disclosed
US-20200309707-A1 REAGENT AND KIT FOR ENHANCING CHEMILUMINESCENT REACTION NATIONAL TAIWAN OCEAN UNIVERSITY (TW) 2020-10-01 US disclosed
US-20070179297-A1 Chemical compounds ASTRAZENECA AB, A SWEDEN CORPORATION 2007-08-02 US disclosed
US-20070179297-A1 Chemical compounds ASTRAZENECA AB, A SWEDEN CORPORATION 2007-08-02 US disclosed
US-7238811-B2 Chemical compounds ASTRAZENECA AB (SE) 2007-07-03 US disclosed
US-7238811-B2 Chemical compounds ASTRAZENECA AB (SE) 2007-07-03 US disclosed
US-7179922-B2 4-Phenyloxypiperidionopiperidine compounds as antiinflammatory agents; autoimmune diseases; rheumatic diseases; cardiovascular disorders ASTRAZENECA AB (SE) 2007-02-20 US disclosed
US-7179922-B2 4-Phenyloxypiperidionopiperidine compounds as antiinflammatory agents; autoimmune diseases; rheumatic diseases; cardiovascular disorders ASTRAZENECA AB (SE) 2007-02-20 US disclosed
WO-2006089700-A1 PYRROLIDINE AND PIPERIDINE ACETYLENE DERIVATIVES FOR USE AS MGLUR5 ANTAGONISTS NOVARTIS AG (CH) 2006-08-31 WO disclosed
EP-0238070-B1 Sulfonylurea compounds, their production and herbicidal use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1993-12-29 EP disclosed
US-5017212-A For rice paddies TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-05-21 US disclosed
EP-0238070-A2 Sulfonylurea compounds, their production and herbicidal use Takeda Chemical Industries, Ltd. (JP) 1987-09-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11112366-B2 Reagent and kit for enhancing chemiluminescent reaction MPO, LPO, KIT RAB9A 3488/4885NPC1 4666/4885KDM4E 822/4885
US-11168083-B2 Inhibitors of Plasma Kallikrein and uses thereof KLKB1, KLK1, KLK5 RAB9A 2329/4885NPC1 2596/4885KDM4E 1766/4885
US-10870638-B2 Pyridazinone compound or its salt, and herbicide containing it H1-0, H1-4, H1-3 RAB9A 2604/4885NPC1 4794/4885KDM4E 1092/4885
US-11136310-B2 Iminotetrahydropyrimidinone derivatives as plasmepsin V inhibitors PEPD, ADAM17, ANPEP RAB9A 3685/4885NPC1 1521/4885KDM4E 2618/4885
US-20230312481-A1 SUBSTITUTED (PHTHALAZIN-1-YLMETHYL)UREAS, SUBSTITUTED N-(PHTHALAZIN-1-YLMETHYL)AMIDES, AND ANALOGUES THEREOF NSD3, PML, NSD1 RAB9A 2543/4885NPC1 910/4885KDM4E 133/4885
US-20070179297-A1 Chemical compounds CCR3, CCR1, CCR4 RAB9A 2189/4885NPC1 887/4885KDM4E 3589/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.