SCHEMBL4340769

SCHEMBL4340769

CC(CC(N)=O)(N[S+]([O-])C(C)(C)C)c1ccc(F)cn1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 1/20 0.33
BACE1 P56817 1/20 0.32
HDAC3 O15379 2/20 0.31
HDAC1 Q13547 2/20 0.31
HDAC2 Q92769 2/20 0.31
HDAC6 Q9UBN7 2/20 0.31
CYP2C19 P33261 1/20 0.31
DGAT1 O75907 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3229309 0.73
SCHEMBL4732409 0.69 CETP (0.56)
SCHEMBL1182281 0.69 CETP (0.56)
SCHEMBL25343042 0.68 KCNN4 (0.39) GABRA5HDAC3HDAC1HDAC2HDAC6
SCHEMBL30087636 0.67 KCNN4 (0.41) GABRA5
SCHEMBL31294557 0.66 DGAT1 (0.40) GABRA5CYP2C19DGAT1CNR1CNR2
SCHEMBL4340774 0.66 APLNR (0.40) HDAC6
SCHEMBL15839715 0.65 HDAC3 (0.39) BACE1HDAC3HDAC1HDAC2HDAC6
SCHEMBL15821573 0.65 HDAC3 (0.39) BACE1HDAC3HDAC1HDAC2HDAC6
SCHEMBL15482879 0.64 SMN1; SMN2 (0.33) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095712-A2 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2009-08-06 WO disclosed