SCHEMBL6230133

SCHEMBL6230133

CC(=O)c1cc(NCc2ccccc2Sc2ccc(NC(=O)CC(C=O)c3cc(NCc4ccccc4Sc4ccc5cccnc5c4)cc(Cl)c3O)cc2)cc(Cl)c1O

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSD P07339 11/20 0.37
HDAC6 Q9UBN7 1/20 0.33
NOTUM Q6P988 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
MMP2 P08253 2/20 0.31
MMP9 P14780 2/20 0.31
P2RY14 Q15391 2/20 0.31
ALOX5 P09917 1/20 0.30
EPHX2 P34913 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6230126 0.87 CTSD (0.44) CTSDHDAC6NOTUMTRPV1
SCHEMBL4347491 0.86 CTSD (0.40) CTSDHDAC6NOTUMTRPV1KDR
SCHEMBL6230128 0.84 CTSD (0.39) CTSDHDAC6NOTUMKDR
SCHEMBL6223808 0.79 CTSD (0.39) CTSDHDAC6NOTUMALOX5EPHX2
SCHEMBL4349874 0.79 GAA (0.33) CTSDHDAC6
SCHEMBL4347648 0.77 GAA (0.38) CTSDHDAC6
SCHEMBL4351090 0.76 LMNA (0.41) CTSD
SCHEMBL4350092 0.74 CTSD (0.38) CTSDHDAC6KDR
SCHEMBL4346923 0.73 SLC6A4 (0.43) CTSDHDAC6MMP2MMP9
SCHEMBL4343453 0.73 SMN1; SMN2 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed