SCHEMBL4350720

SCHEMBL4350720

Nc1ncnc2[nH]cc(-c3cccc(Cl)c3)c12

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
STK4 Q13043 15/20 0.68
STK3 Q13188 15/20 0.68
LRRK2 Q5S007 10/20 0.64
BRAF P15056 1/20 0.53
TNNI3K Q59H18 1/20 0.53
ABL1 P00519 1/20 0.52
EGFR P00533 1/20 0.52
SRC P12931 1/20 0.52
KDR P35968 1/20 0.52
ABL2 P42684 1/20 0.52
MAP4K4 O95819 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12438584 0.83 LRRK2 (0.55) STK4STK3LRRK2ABL1EGFR
SCHEMBL8114068 0.83 ADK (0.49) STK4STK3LRRK2
SCHEMBL4353306 0.83 LRRK2 (0.62) STK4STK3LRRK2MAP4K4
SCHEMBL8107168 0.83 LRRK2 (0.62) STK4STK3LRRK2ABL1SRC
SCHEMBL3787081 0.82 SRC (0.50) STK4STK3LRRK2BRAFTNNI3K
SCHEMBL4787827 0.82 DHFR (0.54) STK4STK3LRRK2MAP4K4
SCHEMBL7021288 0.82 LRRK2 (0.63) STK4STK3LRRK2BRAFTNNI3K
SCHEMBL31301542 0.81 STK4 (1.00) STK4STK3LRRK2
SCHEMBL7013879 0.80 LRRK2 (0.65) STK4STK3LRRK2ABL1EGFR
SCHEMBL8112985 0.80 CCNT1 (0.48) STK4STK3LRRK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070328-A1 MODULATORS OF THE EPIDERMAL GROWTH FACTOR RECEPTOR (EGFR) PATHWAY FOR USE IN THE TREATMENT OR PREVENTION OF SUBSTANCE ABUSE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-06-04 WO disclosed
US-6051577-A TYROSINE INHIBITORS; BONE DISORDERS NOVARTIS AG (CH) 2000-04-18 US disclosed
EP-0888353-A1 NOVEL N-7-HETEROCYCLYL PYRROLO 2,3-D]PYRIDINES AND THEIR USE Novartis AG (CH) 1999-01-07 EP disclosed
WO-1997034895-A1 NOVEL N-7-HETEROCYCLYL PYRROLO[2,3-D]PYRIDINES AND THEIR USE NOVARTIS AG (CH) 1997-09-25 WO disclosed