SCHEMBL4352149

SCHEMBL4352149

CC(C)NC(=O)N(S)c1cccc(F)c1O

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.38
ALB P02768 1/20 0.37
ALDH1A1 P00352 3/20 0.36
HPGD P15428 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PTGES O14684 4/20 0.35
POLB P06746 2/20 0.35
GAA P10253 1/20 0.34
TP53 P04637 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4352165 0.82 ERN1 (0.36) ERN1ALDH1A1POLB
SCHEMBL4341634 0.82 ALDH1A1 (0.40) ALDH1A1HPGDL3MBTL1PTGESPOLB
SCHEMBL4351731 0.78 PTGES (0.36) ERN1ALDH1A1L3MBTL1PTGES
SCHEMBL4347354 0.77 KMT2A (0.46) ALBALDH1A1POLBGAATP53
SCHEMBL4351134 0.75 ERN1 (0.36) ERN1ALDH1A1HPGDL3MBTL1PTGES
SCHEMBL4354007 0.75 NPC1 (0.46) ALDH1A1HPGDGAAHTT
SCHEMBL4350070 0.74 NAAA (0.40) ALDH1A1HPGDHTT
SCHEMBL4358609 0.74 POLB (0.40) ALBALDH1A1HPGDPOLBTP53
SCHEMBL4341747 0.73 TSHR (0.45) ALDH1A1GAAHTTNPSR1
SCHEMBL4344053 0.72 GAA (0.41) ALDH1A1GAAHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110065760-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES AND USE THEREOF JERINI AG (DE) 2011-03-17 US claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
US-20070054904-A1 Phenol derivatives and their use as rotamase inhibitors JERINI AG (DE) 2007-03-08 US claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110065760-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES AND USE THEREOF NR1I3, NR1D1, NR1D2 ERN1 1860/4885ALB 4701/4885ALDH1A1 2565/4885
US-20070054904-A1 Phenol derivatives and their use as rotamase inhibitors NR1I3, NR1D1, NR1D2 ERN1 1686/4885ALB 4431/4885ALDH1A1 2767/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.