SCHEMBL4354386

SCHEMBL4354386

O=C(Nc1ccc(O)c(Cl)c1)N(Cc1ccccc1)C1=COCO1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.41
LMNA P02545 2/20 0.40
UBE2M P61081 5/20 0.40
DCUN1D1 Q96GG9 5/20 0.40
TP53 P04637 1/20 0.40
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 2/20 0.38
BCHE P06276 2/20 0.38
ACHE P22303 2/20 0.38
GAA P10253 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
EGFR P00533 1/20 0.37
ERBB2 P04626 1/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
GSK3B P49841 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347969 0.89 EGFR (0.43) LMNAUBE2MDCUN1D1TP53ALDH1A1
SCHEMBL4359232 0.88 ACHE (0.39) LMNAUBE2MDCUN1D1TP53ALDH1A1
SCHEMBL4359597 0.85 LMNA (0.42) LMNAUBE2MDCUN1D1ALDH1A1MEN1
SCHEMBL4345516 0.83 ALOX15 (0.48) LMNATP53MEN1KMT2AMAPT
SCHEMBL4351294 0.82 ALDH1A1 (0.39) LMNAUBE2MDCUN1D1TP53ALDH1A1
SCHEMBL4342217 0.82 EGFR (0.38) LMNAUBE2MDCUN1D1MAPTGAA
SCHEMBL4347110 0.81 EGFR (0.43) ALDH1A1MEN1KMT2AMAPTGAA
SCHEMBL4355478 0.80 EGFR (0.43) LMNAUBE2MDCUN1D1ALDH1A1MAPT
SCHEMBL4352899 0.80 EGFR (0.41) LMNAUBE2MDCUN1D1ALDH1A1MEN1
SCHEMBL4355633 0.79 PDK1 (0.43) UBE2MDCUN1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed