SCHEMBL4355728

SCHEMBL4355728

O=C(O)N1CCCC12CCC(c1cc(F)cc(F)c1)NC2=O

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 7/20 0.34
OPRM1 P35372 4/20 0.34
KCNH2 Q12809 1/20 0.33
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3592708 1.00 SLC6A9 (0.34) SLC6A9OPRM1KCNH2PSEN1PSEN2
SCHEMBL1273808 0.73 ALDH1A1 (0.35) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL978141 0.72 RIPK1 (0.33)
SCHEMBL1069680 0.72 RIPK1 (0.33)
SCHEMBL3811123 0.71
SCHEMBL549324 0.69 GABRP (0.34)
SCHEMBL4346918 0.66 KDM1A (0.32) SLC6A9
SCHEMBL979115 0.66 KDM1A (0.32) SLC6A9
SCHEMBL11895798 0.66 MEN1 (0.33)
SCHEMBL21225273 0.66 GRIN1 (0.38) SLC6A9OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024358-A1 SUBSTITUTED SPIROCYCLIC CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2009-02-18 EP disclosed
WO-2007133491-A1 SUBSTITUTED SPIROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2007-11-22 WO disclosed