SCHEMBL4359014

SCHEMBL4359014

N#Cc1ccc(OBOc2ccc(C#N)c(C#N)c2)cc1C#N

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOB P27338 9/20 0.49
MAOA P21397 7/20 0.46
CYP19A1 P11511 1/20 0.46
ALDH1A1 P00352 3/20 0.41
HPGD P15428 2/20 0.41
PDE4B Q07343 1/20 0.40
AR P10275 3/20 0.39
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 1/20 0.37
USP2 O75604 1/20 0.37
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1277499 0.82 TRPV4 (0.50) AR
SCHEMBL1869777 0.82 PLA2G7 (0.39) AR
SCHEMBL6110658 0.82 AR (0.43) MAOBALDH1A1ARKDM4EUSP2
SCHEMBL29390509 0.79 CYP19A1 (0.65) MAOBMAOACYP19A1ALDH1A1HPGD
SCHEMBL4581525 0.79 CYP19A1 (0.65) MAOBMAOACYP19A1ALDH1A1HPGD
SCHEMBL1668579 0.79 AR (0.61) ALDH1A1ARKDM4EUSP2
SCHEMBL2017293 0.79 XDH (0.49)
SCHEMBL9472016 0.77 CYP19A1 (0.62) MAOBMAOACYP19A1ALDH1A1HPGD
SCHEMBL1377229 0.77 CYP19A1 (0.62) MAOBMAOACYP19A1ALDH1A1HPGD
SCHEMBL9560109 0.76 MAOB (0.57) MAOBMAOACYP19A1ALDH1A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2072509-A1 1-Aryl-1H-quinoline-2-ones: process for their production and their use as anti-inflammatory agents Bayer Schering Pharma Aktiengesellschaft (DE) 2009-06-24 EP disclosed