SCHEMBL4366803

SCHEMBL4366803

CC(C)(CNC(=O)c1cc(F)cc(F)c1)CNc1c(Nc2cnccn2)c(=O)c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
NFKB1 P19838 1/20 0.36
RAB9A P51151 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TSHR P16473 2/20 0.35
MAPKAPK2 P49137 2/20 0.35
KCNA3 P22001 1/20 0.33
KCNA5 P22460 1/20 0.33
PLK1 P53350 1/20 0.33
ALOX15 P16050 1/20 0.33
CASP1 P29466 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HIF1A Q16665 1/20 0.33
LCK P06239 1/20 0.33
KMT2A Q03164 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6988688 0.83 ABCC9 (0.41) NPC1RAB9ATSHRMAPKAPK2
SCHEMBL6990616 0.83 KMT2A (0.50) NPC1MAPTRAB9ASMN1; SMN2TSHR
SCHEMBL6988211 0.78 POLB (0.40) NPC1MAPTRAB9ANPSR1KMT2A
SCHEMBL4366799 0.77 MAPKAPK2 (0.42) NPC1TP53MAPTNFKB1RAB9A
SCHEMBL4366779 0.77 NPC1 (0.37) NPC1TP53MAPTNFKB1RAB9A
SCHEMBL6991619 0.76 TYK2 (0.37) MAPT
SCHEMBL6990458 0.71 CSF1R (0.44) NPC1MAPTRAB9ATSHRMAPKAPK2
SCHEMBL6991687 0.71 KMT2A (0.42) NPC1RAB9ASMN1; SMN2TSHRKMT2A
SCHEMBL6989487 0.70 ALDH1A1 (0.49) RAB9ASMN1; SMN2TSHRKMT2AKDM4E
SCHEMBL6988180 0.69 NAMPT (0.51) NPC1MAPTRAB9ASMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO disclosed
EP-1358160-A1 AMINAL DIONES AS POTASSIUM CHANNEL OPENERS Abbott Laboratories (US) 2003-11-05 EP disclosed
WO-2002062761-A1 AMINAL DIONES AS POTASSIUM CHANNEL OPENERS ABBOTT LABORATORIES (US) 2002-08-15 WO disclosed