SCHEMBL43673

SCHEMBL43673

O=C(CI)ON1C(=O)CCC1=O

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PSMB8 P28062 2/20 0.33
MGLL Q99685 2/20 0.33
PSMB5 P28074 1/20 0.32
ALOX12 P18054 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA2B P29275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL668588 0.88
SCHEMBL2608502 0.83 LMNA (0.34) PSMB8MGLLPSMB5
SCHEMBL2618714 0.82 MGLL (0.34) PSMB8MGLLPSMB5ALOX12ADORA3
SCHEMBL43576 0.82 PSMB8 (0.35) PSMB8MGLLPSMB5ALOX12ADORA3
SCHEMBL1603240 0.80 KMT2A (0.33) PSMB8MGLLPSMB5ALOX12
SCHEMBL3805679 0.80 MGLL (0.33) PSMB8MGLLPSMB5ALOX12ADORA3
SCHEMBL31522720 0.80 PSMB8 (0.34) PSMB8MGLLPSMB5ALOX12ADORA3
SCHEMBL14706629 0.80 PSMB8 (0.31) PSMB8PSMB5
SCHEMBL21342214 0.80 MGLL (0.31) MGLL
SCHEMBL1140516 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3784 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4749282-A2 HOMOGENOUS IMMUNOASSAY WITH COMPENSATION FOR BACKGROUND SIGNAL IDEXX Laboratories, Inc. (US) 2026-05-27 EP claimed
CN-115581847-B Photodynamic balloon catheter system 杭州矩正医疗科技有限公司 2026-05-19 CN claimed
EP-4713024-A1 CONJUGATE AND THE PREPARATION THEREOF Nanjing University (CN) 2026-03-25 EP claimed
US-20260043066-A1 COMPOSITIONS AND METHODS RELATED TO KETHOXAL DERIVATIVES THE UNIVERSITY OF CHICAGO (US) 2026-02-12 US claimed
US-20260035410-A1 THERAPEUTIC PEPTIDES AND METHODS OF PEPTIDE DESIGN WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2026-02-05 US claimed
US-12516150-B2 Organic solvent-soluble copolymer polyester, composition for forming ultrafiltration membrane comprising same, and high water permeability reverse osmosis membrane prepared therefrom TORAY ADVANCED MATERIALS KOREA INC. (KR) 2026-01-06 US claimed
US-12472267-B2 Compositions containing nucleic acid nanoparticles with modular functionality Sixfold Bioscience Ltd. (GB) 2025-11-18 US claimed
US-12428477-B2 Antibody-drug conjugates comprising anti-TM4SF1 antibodies and methods of using the same ANGIEX, INC. (US) 2025-09-30 US claimed
US-20250195679-A1 ANTIBODY-DRUG CONJUGATE AND USE THEREOF SHANGHAI HUAOTA BIOPHARMACEUTICAL CO., LTD. (CN) 2025-06-19 US claimed
EP-4494658-A1 ANTIBODY-DRUG CONJUGATE AND USE THEREOF Shanghai Huaota Biopharmaceutical Co., Ltd. (CN) 2025-01-22 EP claimed
WO-2007083984-A1 CONJUGATE COMPRISING PHARMACEUTICAL ACTIVE COMPOUND COVALENTLY BOUND TO MUCOADHESIVE POLYMER AND TRANSMUCOSAL DELIVERY METHOD OF PHARMACEUTICAL ACTIVE COMPOUND USING THE SAME GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2007-07-26 WO claimed
EP-1689846-A2 METHOD OF TARGETING SPECIFIC CELL POPULATIONS USING CELL-BINDING AGENT MAYTANSINOID CONJUGATES LINKED VIA A NON-CLEAVABLE LINKER, SAID CONJUGATES, AND METHODS OF MAKING SAID CONJUGATES Immunogen, Inc. (US) 2006-08-16 EP claimed
US-20050169933-A1 Method of targeting specific cell populations using cell-binding agent maytansinoid conjugates linked via a non-cleavable linker, said conjugates, and methods of making said conjugates IMMUNOGEN, INC. 2005-08-04 US claimed
WO-2005037992-A2 METHOD OF TARGETING SPECIFIC CELL POPULATIONS USING CELL-BINDING AGENT MAYTANSINOID CONJUGATES LINKED VIA A NON-CLEAVABLE LINKER, SAID CONJUGATES, AND METHODS OF MAKING SAID CONJUGATES IMMUNOGEN, INC. (US) 2005-04-28 WO claimed
EP-0977588-B1 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES JACKSON H M FOUND MILITARY MED (US) 2004-10-06 EP claimed
US-6613894-B1 Bonding the nucleoside to a solid support, deprotecting using an acid, reacting with a nucleoside phosphoramidite; oxidizing and coupling a biomolecule to the product NANOGEN RECOGNOMICS GMBH (DE) 2003-09-02 US claimed
US-6160128-A Tritioacetylating reagents and processes for preparation thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2000-12-12 US claimed
US-6087328-A FUNCTIONALIZING A POLYSACCHARIDE WITH ONE OR MORE PENDANT HALOACYL GROUPS, THEN THE FUNCTIONALIZED GROUP IS REACTED WITH PROTEIN OR PEPTIDE TO FORM A COVALENTLY LINKED CONJUGATE, USEFUL AS A VACCINE AGAINST BACTERIA, FUNGI OR VIRUSES HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE (US) 2000-07-11 US claimed
EP-0977588-A2 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE (US) 2000-02-09 EP claimed
WO-1998047530-A2 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE (US) 1998-10-29 WO claimed