SCHEMBL4371077

SCHEMBL4371077

CNC(=O)Cc1ccccc1O

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.61
HSPA5 P11021 1/20 0.52
TSHR P16473 2/20 0.52
HIF1A Q16665 2/20 0.52
CYP2D6 P10635 1/20 0.52
CA12 O43570 6/20 0.48
CA2 P00918 6/20 0.48
MAPT P10636 2/20 0.47
CA9 Q16790 5/20 0.47
KDM4E B2RXH2 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
ATM Q13315 1/20 0.45
MPO P05164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10203654 0.83 AKR1B1 (0.50) AKR1B1HSPA5TSHRHIF1ACYP2D6
SCHEMBL8569167 0.82 GABRA1 (0.41) TSHRCYP2D6ATM
SCHEMBL3068210 0.81 HSPA5 (0.48) AKR1B1HSPA5TSHRHIF1ACYP2D6
SCHEMBL3860837 0.81 AKR1B1 (0.57) AKR1B1HSPA5TSHRHIF1ACYP2D6
SCHEMBL28209919 0.81 AKR1B1 (0.57) AKR1B1HSPA5TSHRHIF1ACYP2D6
SCHEMBL5298485 0.80 NPC1 (0.54)
SCHEMBL22275806 0.80 GLS (0.47) CYP2D6ATM
SCHEMBL5738109 0.80 AKR1B1 (0.61) AKR1B1HSPA5TSHRHIF1ACYP2D6
SCHEMBL22316652 0.78 KMT2A (0.45) TSHRMAPTKDM4ESIGMAR1ATM
SCHEMBL20918037 0.78 CYP1A2 (0.39) TSHRCYP2D6MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4249480-A1 DIPHENYLPYRAZOLE COMPOUND, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Northwest A&F University (CN) 2023-09-27 EP disclosed
EP-4070795-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME Salk Institute for Biological Studies (US) 2022-10-12 EP disclosed
EP-3185868-B1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME SALK INST FOR BIOLOGICAL STUDI (US) 2022-04-06 EP disclosed
US-10774092-B2 ULK1 inhibitors and methods using same SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2020-09-15 US disclosed
US-10774092-B2 ULK1 inhibitors and methods using same SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2020-09-15 US disclosed
US-10689397-B2 ULK1 inhibitors and methods using same SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2020-06-23 US disclosed
US-10689397-B2 ULK1 inhibitors and methods using same SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 2020-06-23 US disclosed
US-20190284207-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME SALK INSTITUTE FOR BIOLOGICAL STUDIES 2019-09-19 US disclosed
US-20190284207-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME SALK INSTITUTE FOR BIOLOGICAL STUDIES 2019-09-19 US disclosed
US-20190248806-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME SALK INSTITUTE FOR BIOLOGICAL STUDIES 2019-08-15 US disclosed
CN-1906200-A Novel compounds ASTRAZENECA AB (SE) 2007-01-31 CN disclosed
EP-1687311-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2006-08-09 EP disclosed
WO-2005049620-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2005-06-02 WO disclosed
EP-0923539-B1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK AS (DK) 2002-06-05 EP disclosed
EP-1184370-A2 Compounds with growth hormone releasing properties NOVO NORDISK A/S (DK) 2002-03-06 EP disclosed
US-6274584-B1 PEPTIDE DERIVATIVES; BIOAVAILABILITY; ENZYME RESISTANCE; MILK AND WOOL PRODUCTION NOVO NORDISK A/S (DK) 2001-08-14 US disclosed
US-6127354-A FOR TREATMENT OF GROWTH DISORDERS OR TO STIMULATE PRODUCTION OF WOOL OR MILK NOVO NORDISK A/S (DK) 2000-10-03 US disclosed
US-5922770-A NOVEL COMPOUNDS THAT STIMULATE THE RELEASE OF GROWTH HORMONE FROM THE PITUITARY NOVO NORDISK A/S (DK) 1999-07-13 US disclosed
EP-0923539-A1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK A/S (DK) 1999-06-23 EP disclosed
WO-1998003473-A1 COMPOUNDS WITH GROWTH HORMONE RELEASING PROPERTIES NOVO NORDISK A/S (DK) 1998-01-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10689397-B2 ULK1 inhibitors and methods using same ULK1, ULK2, ULK3 AKR1B1 4236/4885HSPA5 929/4885TSHR 4336/4885
US-20190248806-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME ULK1, ULK2, ULK3 AKR1B1 4152/4885HSPA5 901/4885TSHR 4394/4885
US-10774092-B2 ULK1 inhibitors and methods using same ULK1, ULK2, ULK3 AKR1B1 4236/4885HSPA5 929/4885TSHR 4336/4885
US-20190284207-A1 NOVEL ULK1 INHIBITORS AND METHODS USING SAME ULK1, ULK2, ULK3 AKR1B1 4152/4885HSPA5 901/4885TSHR 4394/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.