SCHEMBL437141

SCHEMBL437141

Cc1[nH]c2ccnc(Cl)c2c1C

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.51
BRD4 O60885 5/20 0.41
EGFR P00533 7/20 0.38
BRD2 P25440 4/20 0.38
BRD3 Q15059 4/20 0.38
ABL1 P00519 2/20 0.36
ABL2 P42684 2/20 0.36
AHR P35869 1/20 0.35
PRKCA P17252 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HIF1A Q16665 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14630116 0.83 BRD4 (0.40) SMN1; SMN2BRD4BRD2BRD3KDM4E
SCHEMBL14601904 0.77 SMN1; SMN2 (0.47) SMN1; SMN2EGFRABL1ABL2AHR
SCHEMBL438559 0.74 BRD4 (0.36) SMN1; SMN2BRD4BRD2BRD3KDM4E
SCHEMBL438267 0.74 CCNB2 (0.39) SMN1; SMN2KDM4E
SCHEMBL4909751 0.73 TYMS (0.48)
SCHEMBL31145933 0.73 TP53 (0.49) SMN1; SMN2BRD4BRD2BRD3KDM4E
SCHEMBL31145887 0.71 PTGS2 (0.41) KDM4E
SCHEMBL435783 0.71 MAPT (0.38) SMN1; SMN2BRD4BRD2BRD3KDM4E
SCHEMBL1895093 0.71 EGFR (0.55) EGFRABL1ABL2PRKCA
SCHEMBL1737822 0.69 MAPT (0.47) SMN1; SMN2AHRKDM4EHIF1ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8513277-B2 Pyrrolo[3,2-C] pyridine derivatives and processes for the preparation thereof YUHAN CORPORATION (KR) 2013-08-20 US disclosed
US-8148529-B2 Pyrrolo[3,2-C] pyridine derivatives and processes for the preparation thereof YUHAN CORPORATION (KR) 2012-04-03 US disclosed
US-20120065224-A1 PYRROLO[3,2-C) PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2012-03-15 US disclosed
EP-1784402-B1 PYRROLO[3,2-c]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP (KR) 2011-08-03 EP disclosed
US-20090005409-A1 Pyrrolo[3,2-C] Pyrdine Derivatives and Processes for the Preparation Thereof YUHAN CORPORATION (KR) 2009-01-01 US disclosed
EP-1784402-A1 PYRROLO[3,2-c]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF Yuhan Corporation (KR) 2007-05-16 EP disclosed
WO-2007001139-A1 A COMPOSITION FOR TREATING OR PREVENTING A CANCER COMPRISING PYRROLOPYRIDINE DERIVATIVES YUHAN CORPORATION (KR) 2007-01-04 WO disclosed
WO-2006025714-A1 PYRROLO[3,2-c]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2006-03-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090005409-A1 Pyrrolo[3,2-C] Pyrdine Derivatives and Processes for the Preparation Thereof ATP6AP1, PPOX, PGA5 SMN1; SMN2 4059/4885BRD4 1538/4885EGFR 4570/4885
US-20120065224-A1 PYRROLO[3,2-C) PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF PGA5, ATP6AP1, HPD SMN1; SMN2 3880/4885BRD4 785/4885EGFR 4192/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.