SCHEMBL4374076

SCHEMBL4374076

CC(C)(C)C(NC(=O)O)[C@H](Cc1ccc(Cl)cc1Cl)NC(=O)c1cc(Br)cs1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41
HDAC8 Q9BY41 4/20 0.39
AKT3 Q9Y243 8/20 0.38
MET P08581 1/20 0.37
KIT P10721 1/20 0.37
PRKCA P17252 1/20 0.37
PRKACA P17612 1/20 0.37
PRKACG P22612 1/20 0.37
PRKACB P22694 1/20 0.37
MAPK3 P27361 1/20 0.37
AKT1 P31749 1/20 0.37
AKT2 P31751 1/20 0.37
CAMK2A Q9UQM7 1/20 0.37
GAA P10253 2/20 0.36
EPHX1 P07099 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4562968 1.00 ALDH1A1 (0.41) ALDH1A1LMNAHDAC8AKT3MET
SCHEMBL4378945 0.87 ALDH1A1 (0.44) ALDH1A1LMNA
SCHEMBL4374524 0.81 ALDH1A1 (0.47) ALDH1A1LMNA
SCHEMBL4583485 0.81 ALDH1A1 (0.47) ALDH1A1LMNA
SCHEMBL4375391 0.81 ALDH1A1 (0.42) ALDH1A1LMNAAKT3AKT1AKT2
SCHEMBL4380618 0.80 ALDH1A1 (0.41) ALDH1A1LMNAAKT3AKT1AKT2
SCHEMBL4373508 0.79 ALDH1A1 (0.42) ALDH1A1LMNAAKT3PRKCAPRKACA
SCHEMBL4376938 0.79 ALDH1A1 (0.44) ALDH1A1LMNAAKT3AKT1AKT2
SCHEMBL4373196 0.78 ALDH1A1 (0.45) ALDH1A1LMNA
SCHEMBL1529597 0.77 AKT3 (0.44) ALDH1A1LMNAHDAC8AKT3MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2117523-A1 INHIBITORS OF AKT ACTIVITY SmithKline Beecham Corporation (US) 2009-11-18 EP disclosed
WO-2008098104-A1 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-08-14 WO disclosed