SCHEMBL4376938

SCHEMBL4376938

CC(C)(C)C(NC(=O)O)[C@H](Cc1ccc(F)cc1)NC(=O)c1cc(Br)cs1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
LMNA P02545 1/20 0.44
ULK1 O75385 1/20 0.35
ACE P12821 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
AKT1 P31749 1/20 0.34
AKT2 P31751 1/20 0.34
AKT3 Q9Y243 1/20 0.34
MME P08473 2/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
CA2 P00918 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HRH3 Q9Y5N1 2/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4373196 0.91 ALDH1A1 (0.45) ALDH1A1LMNASMN1; SMN2MAPTMAPK1
SCHEMBL4374524 0.90 ALDH1A1 (0.47) ALDH1A1LMNASMN1; SMN2NPC1RAB9A
SCHEMBL4583485 0.90 ALDH1A1 (0.47) ALDH1A1LMNASMN1; SMN2NPC1RAB9A
SCHEMBL4373508 0.90 ALDH1A1 (0.42) ALDH1A1LMNASMN1; SMN2AKT1AKT2
SCHEMBL4378945 0.90 ALDH1A1 (0.44) ALDH1A1LMNAACESMN1; SMN2MME
SCHEMBL4383634 0.89 ALDH1A1 (0.41) ALDH1A1LMNAAKT1AKT2AKT3
SCHEMBL4375391 0.84 ALDH1A1 (0.42) ALDH1A1LMNASMN1; SMN2AKT1AKT2
SCHEMBL4371837 0.83 HTR2A (0.40) ALDH1A1LMNAAKT1AKT2AKT3
SCHEMBL4380618 0.81 ALDH1A1 (0.41) ALDH1A1LMNAAKT1AKT2AKT3
SCHEMBL4544057 0.80 ULK1 (0.39) ALDH1A1ULK1AKT1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2117523-A1 INHIBITORS OF AKT ACTIVITY SmithKline Beecham Corporation (US) 2009-11-18 EP disclosed
WO-2008098104-A1 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-08-14 WO disclosed