SCHEMBL4374429

SCHEMBL4374429

NNc1cc(Cl)cc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 3/20 0.53
SLC13A3 Q8WWT9 1/20 0.46
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
P2RX1 P51575 5/20 0.38
P2RX4 Q99571 2/20 0.37
P2RX7 Q99572 2/20 0.37
TMPRSS4 Q9NRS4 2/20 0.37
IKBKB O14920 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4376336 0.98 RAPGEF4 (0.51) RAPGEF4SLC13A3HDAC3HDAC1HDAC2
SCHEMBL998165 0.84 IDO1 (0.46) RAPGEF4MAPTALDH1A1P2RX1P2RX4
Hydrochloric Acid SCHEMBL999258 0.82 IDO1 (0.48) RAPGEF4MAPTALDH1A1P2RX1P2RX4
SCHEMBL12706897 0.79 RAPGEF4 (0.57) RAPGEF4SLC13A3HDAC3HDAC1HDAC2
SCHEMBL997922 0.77 HDAC3 (0.42) RAPGEF4HDAC3HDAC1HDAC2HDAC6
SCHEMBL321756 0.77 AHR (0.52) RAPGEF4SLC13A3HDAC3HDAC1HDAC2
SCHEMBL486657 0.77 IDO1 (0.50) RAPGEF4MEN1KMT2AMAPTALDH1A1
SCHEMBL3786224 0.77 RAPGEF4 (0.47) RAPGEF4SLC13A3MEN1KMT2AALDH1A1
SCHEMBL25112073 0.75 MAPT (0.43) RAPGEF4MAPTALDH1A1SMN1; SMN2P2RX1
SCHEMBL11677821 0.75 RAPGEF4 (0.52) RAPGEF4MAPTALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023036217-A1 ACRYLAMIDE COMPOUND AND USE THEREOF 南京明德新药研发有限公司 2023-03-16 WO disclosed
WO-2009117421-A2 HETEROCYCLIC MODULATORS OF GPR119 FOR TREATMENT OF DISEASE KALYPSYS, INC. (US) 2009-09-24 WO disclosed