SCHEMBL437834

SCHEMBL437834

Cc1[nH]c2ccnc(Cl)c2c1Cc1cccc(F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.45
SNCA P37840 1/20 0.44
ADCY10 Q96PN6 1/20 0.38
ENPP1 P22413 1/20 0.37
POLB P06746 1/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
P2RX7 Q99572 1/20 0.34
NR3C2 P08235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL438267 0.86 CCNB2 (0.39) SLC2A1PTGS1PTGS2TAAR1
SCHEMBL435782 0.78 SLC2A1 (0.38) SLC2A1L3MBTL1PTGS1PTGS2ALDH1A1
SCHEMBL436711 0.74 KDM4E (0.43) POLBL3MBTL1ALDH1A1LMNARAB9A
SCHEMBL441514 0.74 SLC2A1 (0.43) SLC2A1SNCAPTGS1PTGS2PDE3B
Hydrochloric Acid SCHEMBL433810 0.74 KDM4E (0.42) POLBL3MBTL1ALDH1A1LMNARAB9A
SCHEMBL693706 0.72 MAPT (0.50) SLC2A1SNCAPOLBPTGS1PTGS2
SCHEMBL858273 0.72 ENPP1 (0.44) ADCY10ENPP1L3MBTL1ALDH1A1HPGD
SCHEMBL439027 0.70 UTS2R (0.54) L3MBTL1PTGS1PTGS2ALDH1A1HPGD
SCHEMBL855862 0.70 ENPP1 (0.47) ADCY10ENPP1L3MBTL1ALDH1A1LMNA
SCHEMBL438559 0.70 BRD4 (0.36) SLC2A1POLBALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8513277-B2 Pyrrolo[3,2-C] pyridine derivatives and processes for the preparation thereof YUHAN CORPORATION (KR) 2013-08-20 US disclosed
US-8148529-B2 Pyrrolo[3,2-C] pyridine derivatives and processes for the preparation thereof YUHAN CORPORATION (KR) 2012-04-03 US disclosed
US-20120065224-A1 PYRROLO[3,2-C) PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2012-03-15 US disclosed
EP-1784402-B1 PYRROLO[3,2-c]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP (KR) 2011-08-03 EP disclosed
US-20090005409-A1 Pyrrolo[3,2-C] Pyrdine Derivatives and Processes for the Preparation Thereof YUHAN CORPORATION (KR) 2009-01-01 US disclosed
EP-1784402-A1 PYRROLO[3,2-c]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF Yuhan Corporation (KR) 2007-05-16 EP disclosed
WO-2006025714-A1 PYRROLO[3,2-c]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2006-03-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090005409-A1 Pyrrolo[3,2-C] Pyrdine Derivatives and Processes for the Preparation Thereof ATP6AP1, PPOX, PGA5 SLC2A1 3328/4885SNCA 1292/4885ADCY10 2276/4885
US-20120065224-A1 PYRROLO[3,2-C) PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF PGA5, ATP6AP1, HPD SLC2A1 3940/4885SNCA 1285/4885ADCY10 1582/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.