SCHEMBL4378623

SCHEMBL4378623

COc1ccc2c([c]c(C)n2Cc2ccccc2Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 2/20 0.52
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ALOX5AP P20292 1/20 0.45
MAPT P10636 4/20 0.45
F2RL3 Q96RI0 2/20 0.43
PTGER3 P43115 1/20 0.42
OPRM1 P35372 1/20 0.42
RXFP1 Q9HBX9 1/20 0.41
TP53 P04637 4/20 0.41
BRD4 O60885 1/20 0.40
CASR P41180 1/20 0.40
POLB P06746 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15062678 0.86 PLA2G2A (0.43) PLA2G2AMEN1KMT2AMAPTTHRB
SCHEMBL8360274 0.84 ALDH1A1 (0.52) PLA2G2AKMT2AMAPTTP53POLB
SCHEMBL4541878 0.81 ALDH1A1 (0.53) PLA2G2AMEN1KMT2AMAPTPOLB
SCHEMBL4375652 0.81 ALDH1A1 (0.50) PLA2G2AMEN1KMT2AMAPTTP53
SCHEMBL27789954 0.76 CCR2 (0.52) PLA2G2AMEN1KMT2AMAPTTP53
SCHEMBL4381044 0.75 MAPT (0.43) PLA2G2AMEN1KMT2AMAPTTP53
SCHEMBL3088631 0.73 P2RX4 (0.54) MEN1KMT2AMAPTTP53POLB
SCHEMBL11461389 0.73 PLA2G2A (0.58) PLA2G2AMEN1KMT2AMAPTPTGER3
SCHEMBL2071948 0.73 GABRA1 (0.54) MEN1KMT2AMAPTBRD4POLB
SCHEMBL8356890 0.72 PLA2G2A (0.52) PLA2G2AMEN1KMT2AMAPTOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed