SCHEMBL8360274

SCHEMBL8360274

COc1ccc2c([c]c(C)n2Cc2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
HTT P42858 2/20 0.52
POLB P06746 1/20 0.52
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
KMT2A Q03164 1/20 0.51
PLA2G2A P14555 16/20 0.50
PLA2G1B P04054 1/20 0.50
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HTR6 P50406 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4541878 0.92 ALDH1A1 (0.53) ALDH1A1HTTPOLBTSHRMAPK1
SCHEMBL4375652 0.88 ALDH1A1 (0.50) ALDH1A1TSHRMAPK1KMT2APLA2G2A
SCHEMBL2071948 0.85 GABRA1 (0.54) ALDH1A1HTTPOLBTSHRMAPK1
SCHEMBL8356890 0.84 PLA2G2A (0.52) ALDH1A1POLBKMT2APLA2G2AMAPT
SCHEMBL4378623 0.84 PLA2G2A (0.52) POLBKMT2APLA2G2ATP53MAPT
SCHEMBL27789954 0.83 CCR2 (0.52) ALDH1A1HTTTSHRMAPK1KMT2A
SCHEMBL3088631 0.83 P2RX4 (0.54) ALDH1A1HTTPOLBMAPK1KMT2A
SCHEMBL8354114 0.83 ALDH1A1 (0.49) ALDH1A1HTTPOLBTSHRMAPK1
SCHEMBL8356349 0.79 ALDH1A1 (0.46) ALDH1A1HTTPOLBTSHRMAPK1
SCHEMBL10399302 0.79 CYP19A1 (0.48) ALDH1A1HTTTSHRMAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877202-A Indole derivatives useful to treat estrogen-related neoplasms and disorders AVENTISUB II INC. 1999-03-02 US disclosed