SCHEMBL4379039

SCHEMBL4379039

O=C(Nc1ccncc1)Nc1cnccn1.O=C(Nc1cnccn1)Nc1c2c(nc3ccccc13)CCCC2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.53
HTT P42858 2/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 1/20 0.49
PLK4 O00444 1/20 0.48
CHEK1 O14757 1/20 0.48
PDPK1 O15530 1/20 0.48
PRKD3 O94806 1/20 0.48
MAP4K4 O95819 1/20 0.48
CHEK2 O96017 1/20 0.48
CDK1 P06493 1/20 0.48
PIM1 P11309 1/20 0.48
RPS6KB1 P23443 1/20 0.48
CDK2 P24941 1/20 0.48
FLT4 P35916 1/20 0.48
KDR P35968 1/20 0.48
CSNK1D P48730 1/20 0.48
CDK8 P49336 1/20 0.48
CLK2 P49760 1/20 0.48
GSK3A P49840 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3798774 0.94 HTT (0.55) ACHEHTTGAAMAPTPLK4
SCHEMBL4560545 0.86 CHEK1 (0.51) ACHEHTTGAAMAPTPLK4
SCHEMBL4379043 0.84 ACHE (0.50) ACHEHTTGAAMAPTBCHE
SCHEMBL4560546 0.78 HTT (0.43) ACHEHTTGAAMAPTBCHE
SCHEMBL10061487 0.76 HTT (0.67) ACHEHTTGAAMAPTBCHE
SCHEMBL3804620 0.75 RAB9A (0.74) GAA
SCHEMBL10061986 0.74 APP (0.62) ACHEHTTGAAMAPTBCHE
SCHEMBL9208663 0.74 HTT (0.74) ACHEHTTGAAMAPTBCHE
SCHEMBL14517928 0.73 RAB9A (0.72) GAAPIM1PIM3AURKB
SCHEMBL9749208 0.73 HTT (0.64) ACHEHTTGAAMAPTBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091943-A2 HETEROCYCLIC COMPOUNDS AND THEIR USE AS GLYCOGEN SYNTHASE KINASE 3 INHIBITORS Abbott GmbH & Co. KG (DE) 2009-08-26 EP disclosed
WO-2008046919-A2 HETEROCYCLIC COMPOUNDS AND THEIR USE AS GLYCOGEN SYNTHASE KINASE 3 INHIBITORS ABBOTT GMBH & CO. KG (DE) 2008-04-24 WO disclosed