SCHEMBL4379043

SCHEMBL4379043

O=C(Nc1ccncc1)N(c1cnccn1)N(C(=O)Nc1c2c(nc3ccccc13)CCCC2)c1cnccn1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.50
HTT P42858 2/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.48
BCHE P06276 2/20 0.47
HDAC6 Q9UBN7 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4379039 0.84 ACHE (0.53) ACHEHTTGAAMAPTBCHE
SCHEMBL4560546 0.84 HTT (0.43) ACHEHTTGAAMAPTBCHE
SCHEMBL3798774 0.79 HTT (0.55) ACHEHTTGAAMAPTBCHE
SCHEMBL10061487 0.75 HTT (0.67) ACHEHTTGAAMAPTBCHE
SCHEMBL9208663 0.73 HTT (0.74) ACHEHTTGAAMAPTBCHE
SCHEMBL9749208 0.72 HTT (0.64) ACHEHTTGAAMAPTBCHE
SCHEMBL4560545 0.72 CHEK1 (0.51) ACHEHTTGAAMAPTBCHE
SCHEMBL8473136 0.72 HTT (0.69) ACHEHTTGAAMAPTBCHE
SCHEMBL8472225 0.71 HTT (0.71) ACHEHTTGAAMAPTBCHE
SCHEMBL8476129 0.70 HTT (0.73) ACHEHTTGAAMAPTBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091943-A2 HETEROCYCLIC COMPOUNDS AND THEIR USE AS GLYCOGEN SYNTHASE KINASE 3 INHIBITORS Abbott GmbH & Co. KG (DE) 2009-08-26 EP disclosed
WO-2008046919-A2 HETEROCYCLIC COMPOUNDS AND THEIR USE AS GLYCOGEN SYNTHASE KINASE 3 INHIBITORS ABBOTT GMBH & CO. KG (DE) 2008-04-24 WO disclosed