SCHEMBL4383634

SCHEMBL4383634

CC(C)(C)C(NC(=O)O)[C@H](Cc1cccc(F)c1)NC(=O)c1cc(Br)cs1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
PIN1 Q13526 3/20 0.39
SLC1A1 P43005 2/20 0.38
ROCK1 Q13464 3/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
GRM5 P41594 2/20 0.38
CCR1 P32246 3/20 0.37
CHRM2 P08172 1/20 0.37
CCR5 P51681 1/20 0.37
PRKCA P17252 2/20 0.37
AKT1 P31749 2/20 0.37
AKT2 P31751 2/20 0.37
AKT3 Q9Y243 2/20 0.37
EGFR P00533 1/20 0.37
PIM1 P11309 1/20 0.37
SYK P43405 1/20 0.37
MAPKAPK2 P49137 1/20 0.37
GSK3B P49841 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4373196 0.90 ALDH1A1 (0.45) ALDH1A1LMNA
SCHEMBL4583485 0.90 ALDH1A1 (0.47) ALDH1A1LMNACCR1MEN1KMT2A
SCHEMBL4374524 0.90 ALDH1A1 (0.47) ALDH1A1LMNACCR1MEN1KMT2A
SCHEMBL4376938 0.89 ALDH1A1 (0.44) ALDH1A1LMNACTSSCTSKAKT1
SCHEMBL4371837 0.89 HTR2A (0.40) ALDH1A1LMNAPIN1AKT1AKT2
SCHEMBL4373508 0.87 ALDH1A1 (0.42) ALDH1A1LMNAPIN1ROCK1PRKCA
SCHEMBL4375391 0.83 ALDH1A1 (0.42) ALDH1A1LMNACTSSCTSKCCR1
SCHEMBL4378945 0.83 ALDH1A1 (0.44) ALDH1A1LMNAGSK3BPPARGKMT2A
SCHEMBL4544087 0.81 AKT1 (0.39) ROCK1GRM5CCR1CHRM2CCR5
SCHEMBL4380618 0.80 ALDH1A1 (0.41) ALDH1A1LMNAAKT1AKT2AKT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2117523-A1 INHIBITORS OF AKT ACTIVITY SmithKline Beecham Corporation (US) 2009-11-18 EP disclosed
WO-2008098104-A1 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-08-14 WO disclosed