SCHEMBL4384076

SCHEMBL4384076

COc1ccc2c([c]cn2Cc2ccc(Cl)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 2/20 0.46
MAPT P10636 4/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
MEN1 O00255 1/20 0.43
RGS12 O14924 1/20 0.43
PKM P14618 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
MAPK1 P28482 1/20 0.43
GNAI1 P63096 1/20 0.43
PMP22 Q01453 1/20 0.43
KMT2A Q03164 1/20 0.43
HIF1A Q16665 1/20 0.43
TP53 P04637 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29136189 0.92 MAPT (0.47) KCNA3MAPTALDH1A1LMNAMEN1
SCHEMBL2117424 0.87 HTR6 (0.48) KCNA3MAPTALDH1A1LMNATSHR
SCHEMBL29136213 0.84 CCR2 (0.51) MAPTLMNAMEN1TSHRKMT2A
SCHEMBL15062690 0.84 IDO1 (0.39) MAPTLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL4377626 0.81 CACNB4 (0.45) MAPTALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL22632586 0.79 HTR6 (0.43) MAPTALDH1A1MEN1TSHRKMT2A
SCHEMBL3091133 0.78 P2RX4 (0.48) MAPTALDH1A1LMNAMAPK1TP53
SCHEMBL6235287 0.75 GRM2 (0.46) MAPTALDH1A1MEN1TSHRKMT2A
SCHEMBL6087656 0.75 HDAC8 (0.57) KCNA3MAPTLMNATP53CCR2
SCHEMBL29136198 0.75 MAPT (0.46) MAPTALDH1A1LMNAMEN1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2610244-A1 Indole compounds Ironwood Pharmaceuticals, Inc. (US) 2013-07-03 EP disclosed
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed