SCHEMBL4386892

SCHEMBL4386892

CCOc1ccc2c(c1)c(C(=O)C(=O)Nc1ccc(OC)cc1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl.COc1ccc(NC(=O)C(=O)c2c(C(F)(F)F)n(Cc3ccc(Cl)cc3Cl)c3ccc(O)cc23)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
POLB P06746 1/20 0.41
KCNH2 Q12809 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
PLA2G2A P14555 2/20 0.38
FAAH O00519 1/20 0.38
EDNRB P24530 2/20 0.37
MAPK1 P28482 2/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HTT P42858 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HPGD P15428 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
USP2 O75604 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3008455 0.96 MEN1 (0.42) MEN1KMT2APOLBKCNH2NPC1
SCHEMBL2997974 0.95 KCNH2 (0.44) MEN1KMT2AKCNH2NPC1RAB9A
SCHEMBL3010861 0.92 MEN1 (0.44) MEN1KMT2APOLBPLA2G2AFAAH
SCHEMBL2995848 0.91 KMT2A (0.45) MEN1KMT2AKCNH2NPC1RAB9A
SCHEMBL2996462 0.90 KCNH2 (0.45) MEN1KMT2AKCNH2NPC1RAB9A
SCHEMBL3008903 0.89 MEN1 (0.41) MEN1KMT2APOLBEDNRBMAPT
SCHEMBL3008225 0.89 PLA2G2A (0.45) MEN1KMT2AKCNH2NPC1RAB9A
SCHEMBL3002874 0.89 PTGS2 (0.46) PLA2G2AFAAHEDNRBMAPTHTT
SCHEMBL3005046 0.88 FAAH (0.41) MEN1KMT2APOLBFAAHHTT
SCHEMBL3001593 0.88 L3MBTL1 (0.41) MEN1KMT2AFAAHMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed